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N-{imidazo[1,2-a]pyridin-2-ylmethyl}-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
N3-cyclopentyl-1-(3-methylbutyl)-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(1H-indol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(propan-2-yl)propanamide
N-ethyl-5-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-1H-pyrazole-3-carboxamide
3-{1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
3-(5-acetylthiophene-2-carbonyl)-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
3-(4-methylphenoxymethyl)-1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
[(2S,4R)-4-(dimethylamino)-1-(6-ethyl-2-methylquinoline-4-carbonyl)pyrrolidin-2-yl]methanol
3-methoxy-1-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
N-methyl-N-(2-methylpropyl)-4-{thieno[3,2-d]pyrimidin-4-yl}morpholine-2-carboxamide
1-(6-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyridin-3-yl)ethan-1-one
3-benzyl-4-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-N-tert-butyl-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carboxamide
1-[1'-(2-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-4-methoxyphenol
2-(1-{[5-(2-cyanophenyl)furan-2-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
4-[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-1-(thiolan-3-yl)piperidine
4-methyl-6-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-2-amine
[1-(3-methoxyphenyl)ethyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-cyclopropyl-1-{1-[1-(4-fluorophenyl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(methylsulfanyl)pyridine-3-carboxamide
N-(1-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
1-cyclopentanecarbonyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
N-ethyl-N-[2-(morpholin-4-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
4-(3-fluorophenoxy)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
N,N-dimethyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-(2-methoxyethyl)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]propanamide
4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-1-ethyl-3-methylpiperazin-2-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(thiophene-2-carbonyl)-6-azaspiro[2.5]octane
2-methoxy-3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridine
15-methyl-N-[(1-methylpiperidin-3-yl)methyl]-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-(piperidin-1-ylmethyl)-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-ol
3-(2-hydroxyphenyl)-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[(2-fluorophenyl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
methyl 4-{2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-ylmethyl}-1H-pyrazole-3-carboxylate
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-propoxyethan-1-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-propylpyridine-4-carboxamide
7-fluoro-4-{3-[(methylsulfanyl)methyl]piperidin-1-yl}quinazoline
6-methoxy-N-[3-methoxy-4-(3-methylbutanamido)phenyl]hexanamide
2-{6-chloro-3-[(2-methylpiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-ethyl-4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-(3-phenyl-1,2,4-thiadiazol-5-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxamide
1-(4-{[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol