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N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(phenylamino)pyrimidine-5-carboxamide
N-(3,4-dimethoxyphenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amine
3-cyclohexyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
6-(aminomethyl)-2-(3-{[(2-phenylethyl)(propyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]pentane-1,2-dione
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(pyridin-3-ylmethyl)amine
N-cyclopropyl-1-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-4-yl}piperidine-4-carboxamide
1-(3-fluoro-2-methylphenyl)-3-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}urea
7-(2-hydroxyethyl)-2-(2-methyl-1,3-benzothiazole-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(pyridin-4-ylmethyl)-4-{[1-(thiolan-3-yl)piperidin-4-yl]oxy}benzamide
N-[2-(morpholin-4-yl)ethyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
2-[(4-chlorophenyl)methyl]-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
N-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-4-methylbenzamide
3-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
4-methyl-N-(oxolan-2-ylmethyl)-N-{[3-(thiophen-3-ylmethoxy)phenyl]methyl}benzamide
3-({4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}sulfonyl)-N-methylbenzamide
N-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2,3,5,6-tetramethyl-N-[2-(methylamino)ethyl]benzamide
1-[benzyl(methyl)amino]-3-(4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(1S,4S)-2-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
(3R,4S)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-cyclopropylpyrrolidin-3-amine
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[2-(1H-imidazol-1-yl)ethyl]piperidin-4-amine
3-[(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
methyl 4-{2-[(3-fluorophenyl)methyl]morpholine-4-carbonyl}benzoate
N-cyclopropyl-5-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-[2-(3-hydroxyphenyl)ethyl]-N,N-dimethylpiperidine-1-carboxamide
ethyl 3-({3-[benzyl(methyl)carbamoyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl}amino)propanoate
2-(2-chloro-4-{[3-hydroxy-3-(hydroxymethyl)pyrrolidin-1-yl]methyl}-6-methoxyphenoxy)acetamide
2-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
3,5-dichloro-N-(2-ethyl-2,5-dihydroxypentyl)-4-methylbenzamide
N,N-dimethyl-3-({2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}sulfonyl)benzamide
6-methyl-2-{[3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}quinolin-4-ol
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(quinolin-3-ylmethyl)acetamide
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propyl]piperidin-4-ol
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
N-(2-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
9-[(4-chlorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(azepan-1-yl)-3-[3-(azetidin-1-ylmethyl)phenoxy]propan-2-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-6-oxo-N-(oxolan-2-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-(4-{[4-(1-benzofuran-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
N-(1-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-(4-methyl-1H-pyrazol-5-yl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
3-methoxy-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]butan-1-one