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4-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
1-(4-fluorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]cyclopropane-1-carboxamide
3-propyl-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[1-(3-chlorobenzoyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
2-{[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
(2S,4S)-4-amino-1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-propyl-5-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyrimidin-2-amine
3-(1H-imidazol-1-ylmethyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine
[1-(4-methoxy-2-methylbenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
7-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(3R,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]butane-1-sulfonamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3,4-dimethoxyphenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
4-hydroxy-N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N,2-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(2,6-difluoro-3-methylphenyl)methyl]-9-oxa-2-azaspiro[5.5]undecane
2-({1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl}sulfanyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-[(6-chloropyridin-3-yl)methyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
[(2-methyl-1H-imidazol-4-yl)methyl][(2-phenoxypyridin-3-yl)methyl]amine
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
8-chloro-2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}quinoline
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
N-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-(3-chloro-4-fluorophenoxy)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one
N-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(1-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]piperidine-3-carboxamide
2-{4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}pyridine-3-carboxamide
6-methoxy-2-oxo-N-[2-(pyridin-4-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-({[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
9-[2-methyl-2-(morpholin-4-yl)propyl]-3-oxa-9-azaspiro[5.5]undecane
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-cyclopropyl-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-methyl-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
4-(2-fluorobenzoyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
7-(4-chlorophenyl)-2-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-cyclopropanecarbonyl-N-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]azepan-3-amine
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(1,2-oxazol-3-ylmethyl)amine
6-{[3-(pyridin-3-yl)azetidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
7-cyclohexyl-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide