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N-methyl-3-[2-({[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)phenyl]propanamide
N-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-N-methylthian-4-amine
1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
(2S)-2-amino-1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-(1H-imidazol-4-yl)propan-1-one
3-(4-fluorophenyl)-1-(thiophen-3-ylmethyl)pyrrolidine
N-[2-(dimethylamino)ethyl]-4-methanesulfonyl-N-(thiophen-3-ylmethyl)benzamide
(4aR,8aS)-6-[3-(4-fluorophenyl)benzoyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-(3-ethoxypropyl)-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[(4aR,8aR)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
1-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
2-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-3-(trifluoromethyl)benzene-1-sulfonamide
5-ethyl-N-[(1S)-1-(3-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine
5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-1-(3-methylphenyl)-1H-1,2,4-triazole
2-methyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1-benzofuran-5-carboxamide
N-[(2R,3R)-2-(benzyloxy)-1'-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-(4-fluorophenyl)-1-(4-methylphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
2-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carboxamide
(2E)-3-(2,5-difluorophenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}prop-2-en-1-one
(4aS,7aR)-1-(2-hydroxy-3-methylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
7-[2-(1H-imidazol-2-yl)benzoyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(4-ethoxy-3-methylphenyl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]butanamide
4-{[1-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
2-methyl-6-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
3-hydroxy-3-{[(2-methylbutan-2-yl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridazine
[(3S,5R)-1-(2-cyclopropylpyrimidine-5-carbonyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-{1-azabicyclo[2.2.2]octan-3-yl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N,1,3-trimethyl-N-[2-(morpholin-4-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(2E)-2-methylbut-2-en-1-yl]amino}pyrrolidine-2-carboxamide
7-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2,7,8-trimethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide
[3-benzyl-1-(2,3-dihydro-1-benzofuran-7-carbonyl)piperidin-3-yl]methanol
methyl 3-[(3,5-dimethylphenyl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-4,6-bis(propan-2-yl)phenol
ethyl 1-(2-methoxyethyl)-5-[(8-methoxyquinolin-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{2-[1-(3-fluoro-4-methylbenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
(3S,4R)-1-[2-(morpholin-4-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-methoxy-N-(2-{7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
2-[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
9-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
{4-[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}methanamine
1-phenyl-4-[2-(1-propylpiperidin-4-yl)acetyl]piperazin-2-one