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1-(2-methyl-4-{4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepan-1-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
1-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidine
3-[2-oxo-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1,3-thiazolidine-2,4-dione
1,9-dimethyl-4-[3-(1H-pyrazol-4-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
2-({4-[2-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
2-cyclopentyl-1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-imidazole
2-ethoxy-5-{2-[methyl(oxan-2-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
N-(1-methyl-1H-pyrazol-3-yl)-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
4-({[(5-acetylthiophen-3-yl)methyl](methyl)amino}methyl)-1-ethylpyrrolidin-2-one
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-{4-[1-(3,5-dimethylphenyl)piperidin-4-yl]piperazin-1-yl}pyrazine-2-carbonitrile
N-[(1S)-1-[3-(oxan-4-yl)-1-(quinoxalin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
8-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R)-3-(5,8-dimethoxy-4-methylquinolin-2-yl)-2-methylpropan-1-ol
2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
9-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-({4-[4-(2-fluorophenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[3-(piperidin-1-yl)pyridin-2-yl]formamido}acetic acid
1-({4-methyl-5-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
2-(4-ethoxyphenyl)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}pyrrolidin-3-amine
2-(2,3-dimethoxyphenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5,6-dimethylpyrimidin-4-amine
4-cyclobutanecarbonyl-2-[(3-methoxyphenyl)methyl]morpholine
2-amino-4-(2-methoxyquinolin-3-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-{2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidine-3-carboxamide
1-{1-ethyl-5-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propan-1-one
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-hydroxy-2-phenylethan-1-one
5-methyl-1-[(3-methyloxetan-3-yl)methyl]-5-phenylpiperidin-2-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-phenylpiperidin-3-amine
(3S,4S)-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
3-(4-methoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-5-carboxamide
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(1-phenylethyl)urea
N,2,5-trimethyl-N-(quinolin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(1-{2-[2-(3-fluorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
1-cyclopropyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
(5S,9aS,9bS)-5-[5-(methoxymethyl)furan-2-yl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 3-(1,3-benzothiazol-2-ylmethyl)-9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N'-(3-chloro-4-fluorophenyl)-N-[2-(pyridin-3-ylformamido)ethyl]propanediamide
4-(3-methoxybenzoyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(3-methoxypropyl)piperazine
2-ethyl-4-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
1-[1-(4-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-3,3-dimethylurea
5-(8-fluoro-4-oxo-1,4-dihydroquinoline-2-carbonyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide