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2-(2-methoxyethyl)-8-[3-(3-methoxyphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[(4-methoxyphenyl)methyl]acetamide
3-{3-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]propyl}-3,4-dihydroquinazolin-4-one
2-[5-(1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
N,N,4-trimethyl-3-{[(2-methylprop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(2-{7-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-[2-(2,4-dimethylphenoxy)ethyl]-2-{[5-(furan-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-methylacetamide
4-(4-methylpiperazin-1-yl)-6-[2-(trifluoromethoxy)phenyl]pyrimidin-2-amine
1-methyl-6-(pyridin-4-yl)-N-(2,2,2-trifluoroethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})amine
N-cyclopropyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(1S,5R)-6-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(benzyloxy)ethyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanamide
2-(dimethylamino)-N-(1-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-2-phenylethyl)-N-methylacetamide
1-cyclohexyl-N3-methyl-N5-(2-methylpropyl)-4-oxo-N3-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{3-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}acetamide
N-[4-(pyridin-3-yloxy)phenyl]-1-(4,4,4-trifluorobutyl)piperidine-2-carboxamide
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-{1-[2-(4-fluorophenyl)acetyl]pyrrolidin-2-yl}-N-(2-hydroxyethyl)thiophene-2-carboxamide
1-[2-(dimethylamino)ethyl]-N-[(2,6-dimethylpyridin-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
5-[(isoquinolin-5-yloxy)methyl]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2-oxazole-3-carboxamide
5-benzyl-N-methyl-N-[1-(pyridin-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{[4-(2,6-dimethylphenyl)thiophen-2-yl]methyl}piperazine
2-(5-acetylthiophen-3-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-(2-hydroxyethyl)-8-(2-methoxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
ethyl 4-(oxan-2-ylmethyl)-1-(2,4,5-trifluorobenzenesulfonyl)piperidine-4-carboxylate
3-(1H-imidazol-2-yl)-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
7-chloro-1-(2-phenoxyethyl)-3-{[(propan-2-yl)amino]methyl}-1,2-dihydroquinolin-2-one
9-(2-chloropyridine-4-carbonyl)-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
1-(6-methylpyridin-2-yl)-4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
4-[(2-methylphenyl)sulfanyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
8-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-(4-methoxyphenyl)-N-methyl-3-phenylpropanamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylpyrimidine-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(1H-imidazol-4-ylmethyl)-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
2-[(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]benzonitrile
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(3-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
3-(4-fluorophenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-(2-hydroxyethyl)-4-(2-methoxy-6-methylbenzoyl)-1,4-diazepan-6-ol
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
methyl 8-[(3-ethoxy-4-methoxyphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
4-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
5-(2-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one