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1-[2-(adamantan-1-ylformamido)ethyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2,4-dichlorophenyl)-1-(oxan-3-yl)-1H-imidazole
ethyl 1,5-dibenzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N2,N2-dimethyl-N3-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrazine-2,3-diamine
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine
N-(dimethyl-1,2-oxazol-4-yl)-4-(pyrazin-2-yl)piperazine-1-carboxamide
N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4-methylphenyl)ethan-1-one
ethyl 1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5,6-dimethyl-2-{2-oxo-2-[2-(2-phenylethyl)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
2-ethyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrimidine
5-({[(3-{2-[4-(3-chloro-2-methylbenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
N-[(2-chlorophenyl)methyl]-3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)propanamide
5-(3-fluoro-4-methoxyphenyl)-N-(2-methoxyethyl)furan-2-carboxamide
2-{4-[3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propanamido]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
6-[(3-methoxyphenyl)methoxy]-4-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
2-(4-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
2-cyclopentyl-9-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-2-methyl-4-{[(1S)-1-phenylethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
2-methoxy-1-[1'-(5-propyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(4aR,7aS)-1-benzyl-4-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(morpholin-4-yl)propanamide
1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
1-methyl-1-{2-oxo-2-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}urea
(3R,4S)-4-cyclopropyl-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-amine
N-(1-phenylethyl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-cyclohexyl-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-[methyl(phenyl)amino]ethan-1-one
3-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1-(2,4,6-trimethylpyridin-3-yl)urea
(1S,6R)-9-(morpholine-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)-3-(pyridin-2-yl)propan-1-one
2-(4-{[2-(3-hydroxypropyl)piperidin-1-yl]methyl}phenyl)-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
(3S,4R)-1-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[(2,6-difluorophenyl)methyl]-4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(pyrrolidin-1-yl)pyridazine
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
(2S,4R)-4-[(1-benzylpiperidin-4-yl)amino]-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N,2-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1,6-dimethyl-N-[1-(piperidin-1-ylmethyl)cyclohexyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(pyridin-2-yl)-7-(pyrrolidine-1-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(3,4-dimethoxyphenyl)methyl]-N-(oxan-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-[(3S,4R)-1-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetyl}-4-propylpyrrolidin-3-yl]acetamide
(1S,3R)-N1-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
ethyl 1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(3S,4S)-3-hydroxy-N,N-dimethyl-4-(naphthalen-2-yl)piperidine-1-carboxamide
3-{2-oxo-2-[2-(thiophen-2-yl)azetidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
4-{[4-(2,4-difluoro-3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}pyridine