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methyl 2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
2-(dimethyl-1,2-oxazol-4-yl)-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
2-amino-4-(2-aminopyrimidin-5-yl)-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
(3S,4R)-3-ethyl-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-methylpiperidin-4-ol
1-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
4-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)morpholine
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-b]pyridazine-3-carboxamide
1-cyclohexanecarbonyl-N-(3,4-dimethylphenyl)piperidin-3-amine
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanesulfonamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{1-oxaspiro[4.4]nonan-3-yl}-3-(1H-pyrazol-1-yl)benzamide
7-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,3-diazepane-2,4-dione
3-{5-[5-(hydroxymethyl)furan-2-yl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-ethyl-1-[(4-fluoro-3-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
4-(cyclobutylsulfamoyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}benzamide
(3R,5R)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-(4-fluorophenyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-amine
4-(2,3-dihydro-1H-isoindole-2-sulfonyl)-N-[(2R)-oxolan-2-ylmethyl]benzamide
4-{3-[4-(hydroxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidin-2-yl]methanol
2-(4-{5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-1,2,4-oxadiazol-3-yl}phenyl)ethan-1-ol
N-(1,2-oxazol-3-ylmethyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-cyclohexylacetyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
6-methyl-2-[4-({methyl[(5-phenyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-1'-[(2-hydroxy-3-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
5-(5-methylfuran-2-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2,4-triazin-3-amine
(1S,5R)-3-{[3-(2-hydroxyethoxy)phenyl]methyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
7-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-4-hydroxy-3-methylbenzamide
2-[(4-methoxyphenyl)methyl]-4-[3-(methylsulfanyl)propyl]morpholine
2-(1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}azetidin-3-yl)-1H-1,3-benzodiazole
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-methoxyethyl)piperazine
[4-(2,4-dimethoxyphenyl)pyridin-2-yl]methanol
2-methyl-N-[3-(methylsulfanyl)propyl]-1-benzofuran-5-carboxamide
4,5-dimethyl-6-(1H-pyrazol-3-yl)-2-(pyrrolidin-1-yl)pyrimidine
methyl 2-(cyclohexylsulfamoyl)-6-(pyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-ethyl-8-(propan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
5-(3-chloro-4-propoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
8-[(2S)-2-amino-2-cyclopropylacetyl]-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(adamantan-1-yl)-2-[(pyrimidin-4-yl)amino]ethan-1-ol
methyl (2R)-2-({2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanoate
8-(1-methyl-1H-pyrazole-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide