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3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine
5-methyl-N-[(1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
2-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]urea
(1R,2S,4R)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-(2-ethoxybenzoyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
methyl 3-[4-({methyl[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoate
1-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}naphthalen-2-ol
3-{4-[(2-cyclohexylpyrimidin-5-yl)methyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclohexanecarboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]propanamide
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
ethyl 4-benzyl-1-[(3-methylquinoxalin-2-yl)methyl]piperidine-4-carboxylate
(1S,5R)-3-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}piperidin-2-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
2-cyclopropyl-4-hydroxy-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
1-(2-methylpyridin-4-yl)-4-[4-(pyrrolidin-1-yl)benzoyl]-1,4-diazepane
2-methyl-4-{4-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]phenyl}butan-2-ol
3-[1-(5-fluoro-1,3-dimethyl-1H-indol-2-yl)-N-methylformamido]-N-methylbutanamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
4-[5-(5-methoxy-1H-indol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
N-(2-phenoxyethyl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 2-[(prop-2-en-1-yl)sulfamoyl]-6-[4-(trifluoromethyl)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-({1-[(3,5-dichloro-2-methoxyphenyl)methyl]piperidin-3-yl}methyl)morpholine
2-methyl-4-{3-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]phenyl}butan-2-ol
6-[(4-benzylpiperidin-1-yl)methyl]-2-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[(3-chlorophenyl)methyl]-5-[3-(pyrrolidin-1-yl)butyl]-1H-1,2,4-triazole
2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]-7-methoxy-4-methylquinazoline
ethyl 1-[2-(cyclohex-1-en-1-yl)acetyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-2-hydroxy-4-(methylsulfanyl)butan-1-one
(1S,5R)-6-(pent-2-yn-1-yl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(morpholin-4-yl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)propanamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[3-(propan-2-yl)-1H-pyrazol-5-yl]methyl}amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-[4-(3-hydroxypropyl)piperazin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
(1S,5R)-3-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
[1-(1H-imidazol-1-yl)butan-2-yl](pentan-3-yl)amine
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)piperidine-4-carboxamide
4-{[5-({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}sulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine
4-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-3-yl}-5-phenyl-2-(pyridin-4-yl)pyrimidine
2-[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetic acid
N-[(8-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-2-methylpropanamide
9-[(3,4-dimethylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-hydroxyphenyl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(pyridin-3-ylmethyl)acetamide