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N-[1-(2-methylpropyl)cyclopropyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(dimethylamino)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-methylphenyl)acetamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-(4-methylpiperazin-1-yl)-6-(quinolin-6-yl)pyrimidin-2-amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-({5-[1-(2-methoxyethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-methyl-4-{4-[(2-methylpyrrolidin-1-yl)methyl]phenyl}butan-2-ol
dimethyl({4-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]phenyl}methyl)amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
4-[1-(2-benzyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]pyridine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-ethylpyrimidine-5-carboxamide
2-{4-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]pyrimidin-5-yl}acetic acid
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(2,4-difluorophenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1,2-oxazole-3-carboxamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
4,4,4-trifluoro-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]butanamide
N-[2-(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
N,N-dimethyl-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-sulfonamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(4-fluorophenyl)methyl]-1-phenylpiperazin-2-one
2-{[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl](methyl)amino}-N-methylacetamide
1-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-methyl-N-{2-[4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}methanesulfonamide
methyl 4-{[1-(cyclohexylmethyl)piperidin-3-yl]carbamoyl}butanoate
3-[1-(5-acetylthiophene-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(3S,4S)-1-{3-carbamoyl-5H,6H,7H-cyclopenta[b]pyridin-2-yl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
({2-methoxy-5-[4-(1H-pyrazol-5-yl)phenyl]phenyl}methyl)(methyl)amine
(4S)-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1,3-oxazolidin-2-one
2-(4-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}morpholin-3-yl)-N,N-dimethylacetamide
(3aR,6aS)-5-methyl-N-(2-methylquinolin-8-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
(3R,4R)-3,4-dimethyl-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-ol
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]propanamide
1-(3-fluorophenyl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
1-[(4aR,8aR)-7-[1-(2-fluorophenyl)piperidin-4-yl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
methyl (2S)-2-[3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamido]-3-methylbutanoate
8-(1H-indol-3-ylmethyl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-({[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
2-[2-(1H-imidazol-1-yl)ethyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
(3aS,6aS)-2-cyclohexyl-5-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(1,4-dioxane-2-carbonyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
dimethyl[2-(2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenoxy)ethyl]amine
3-(pyrrolidine-1-carbonyl)-1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]piperidine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-[(4-methylphenyl)methyl]piperidin-3-yl]propanoate
2-(2,3-dihydro-1-benzofuran-7-yl)-6-fluorobenzamide
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-one
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)piperidine-4-carboxamide