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3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyridine
7-(1-benzothiophen-3-yl)-4-(5-methyl-1,3-oxazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(pyridin-3-yl)acetamide
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(1-methyl-1H-indol-4-yl)methyl]pyrrolidin-3-yl]methanol
(3S,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-methyl-4-({2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1H-pyrrole-2-carbonitrile
2-{[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
ethyl 2-{1-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)sulfonyl]piperidin-2-yl}acetate
2-methyl-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-4-carboxylic acid
2-(dimethylamino)-N-(1-ethoxy-2-methylpropan-2-yl)-2-(2-methylphenyl)acetamide
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amine
9-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
5-benzyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(4-methylphenyl)piperazin-2-one
4-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-2,1,3-benzoxadiazole
7-(2,3-dihydro-1-benzofuran-5-carbonyl)-3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
1-{1-methyl-3-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-5-yl}piperidine
1-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
(4aR,7aS)-1-{2-[(2-methoxyethyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
6-[(3-fluorophenyl)methoxy]-4-(1-methylpiperidine-4-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
(3aS,6aS)-2-ethyl-1-oxo-5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethoxy]ethan-1-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-chloropyridazin-3-yl)piperidin-3-ol
N-methyl-2-(morpholine-4-carbonyl)-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-5,6-dimethylthieno[2,3-d]pyrimidine
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-fluorophenyl)ethan-1-one
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-phenylprop-2-yn-1-yl)-N-propylacetamide
N-benzyl-5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]furan-2-carboxamide
N-(2-methoxy-5-methylphenyl)-2-[(1-propylpiperidin-4-yl)amino]acetamide
1-(4-phenyl-1,4-diazepan-1-yl)-2-(1H-pyrazol-1-yl)butan-1-one
3-[(3-chlorophenyl)methyl]-1-ethyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(2-phenylacetamido)pyrrolidin-1-yl]acetic acid
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
3-(2-methoxyethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
2-({4-phenyl-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}methyl)morpholine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylpropan-1-one
4-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-4-oxobutane-1-sulfonamide
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-5-methylpyridine-3-carboxamide
methyl 2-(1-{1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
methyl 3-acetamido-5-{[(3-fluorophenyl)methyl]amino}-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-[(2E)-but-2-en-1-yl]-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,3,4-oxadiazole-2-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
3-({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)amino)-N-methylbutanamide
(1R,5R)-6-(1-benzofuran-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
5-acetyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}thiophene-2-carboxamide
N-(1H-imidazol-4-ylmethyl)-2-[(1-methylpiperidin-4-yl)oxy]aniline
1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione