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1-(5-methyl-2-phenylfuran-3-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
2-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indole
6-(2-chlorophenyl)-N-[1-(pyridin-4-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(2-fluorobenzenesulfonyl)-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-6-phenylpyridazine
6-chloro-2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}imidazo[1,2-a]pyrimidine
ethyl 4-{1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}piperazine-1-carboxylate
N-(cyclopropylmethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-fluoro-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-5-sulfamoylbenzamide
2-(5-acetylthiophen-3-yl)-N-[3-(furan-2-yl)propyl]acetamide
3-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}propan-1-ol
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(3-methoxybenzoyl)piperazine
4-(5-chloro-2-methoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidine
1-(4-{2-methoxy-4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
1-[2-(difluoromethoxy)benzoyl]-3-(piperidin-1-ylmethyl)piperidine
7-fluoro-3-methyl-N-[1-(pyridin-4-yl)propyl]-1-benzofuran-2-carboxamide
1-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-3-ethylpiperidin-3-ol
ethyl 1-(5-cyano-2-hydroxyphenyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
2-{2-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenoxymethyl}pyridine
2-cyclopentyl-9-[2-(1H-imidazol-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({4-[1-(dimethylamino)ethyl]phenyl}methyl)methylamine
N,1-dimethyl-2-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazolidine-4-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethyl-1H-1,2,4-triazole
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-(3-methoxyphenyl)acetamide
N-(2-{4-[(2-methoxy-2-phenylacetamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)benzamide
N-cyclopropyl-1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-4-carboxamide
2-(1-methyl-1H-pyrazole-5-carbonyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N,N-dimethyl-3-[2-({[2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)phenyl]propanamide
2-{2-[(4-methylphenyl)carbamoyl]acetyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-ethoxyphenol
(2S)-2-[2-(2-fluoro-5-methoxyphenyl)-1H-imidazol-1-yl]-3-phenylpropanamide
methyl 2-[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]benzoate
6-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-3-phenylpyrazolo[1,5-a]pyrimidine
3-(pyrazin-2-yl)-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)propan-1-one
1-methoxy-8-[(8-methoxyquinolin-2-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
7-methyl-4-{2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-[2-fluoro-5-(trifluoromethyl)phenyl]-1-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}urea
5-{6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl}benzoic acid
1-[2-(3-chlorophenyl)-2-hydroxyacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(oxolan-3-yl)-5-[4-(propan-2-yloxy)phenyl]-1,2,4-oxadiazole
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
(4aR,7aS)-N,N-dimethyl-4-(6-methylpyridine-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-(pyrazin-2-yl)propan-1-one
4-(2H-1,3-benzodioxol-5-yl)-2-methyl-5-propylpyrimidine