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N-(2,2-difluoroethyl)-4-{[1-(1H-imidazol-2-yl)ethyl]sulfamoyl}benzamide
{3-[(3-chlorophenyl)methyl]-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}methanol
N-{4-[(2,6-dimethylphenyl)carbamoyl]phenyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-({[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
(2S,4R)-4-amino-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
5-(1-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)-3,4-dihydro-1,2,3-benzotriazin-4-one
6-(2,5-dimethylfuran-3-yl)-N-(2-hydroxy-3-methoxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylfuran-2-yl)methyl]amine
2-[5-(2-methyl-6-propylpyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
4-(2,3-dimethoxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
(3aR,6aR)-2-methanesulfonyl-N-methyl-N-(2-phenylethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N,N,4-trimethyl-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-cyclopentyl-2-(2-phenylethyl)morpholine
2,3,5-trimethyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1,2-oxazinan-2-yl)propanamide
(2S,4S)-4-{2-[(dimethylcarbamoyl)amino]acetamido}-N-ethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
2-[3-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)phenoxy]acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
1-(2-ethoxyphenyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
5-(1-cyclopentyl-1H-imidazol-2-yl)-2-(2-methylphenyl)pyrimidine
1-cycloheptyl-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
4-(3,4-diethoxyphenyl)-1H-imidazole
N-ethyl-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-amido)piperidine-1-carboxamide
N-[(3S,4R)-1-(2-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]acetamide
1-(4-{2-[4-(2-ethoxyethyl)piperazin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
6-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinoline
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
4-(2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-2-yl}ethyl)phenol
2-[1-(4-methylpyridin-3-yl)-1H-pyrazol-3-yl]pyrazine
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
4-(3-fluorophenoxy)-1-(oxan-4-yl)piperidine-4-carboxylic acid
3-methyl-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-2-carboxamide
2-[3-(3-methoxyphenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[(3S,4S)-3-hydroxy-4-[methyl(pyridin-3-ylmethyl)amino]pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-{[3-(4-fluorophenoxy)azetidin-1-yl]methyl}-2-methyl-1H-imidazole
3-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroquinolin-2-one
4-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]-1λ6-thiomorpholine-1,1-dione
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
8-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1-(2-hydroxyethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-(2-methyl-1-benzofuran-5-yl)-1H-indazole-3-carboxamide
(2R)-2-amino-2-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
(1S,5R)-3-[(2-chloro-5-fluorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one