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N-[(2-fluorophenyl)methyl]-2-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(2-ethyl-4-methyl-1H-imidazol-5-yl)oxan-4-yl]acetamide
1-(1-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}piperidin-4-yl)pyrrolidin-2-one
{[(3S,4R)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyridin-2-amine
N-[2-(3-methoxyphenyl)-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-(cyclohex-3-en-1-yl)-1-[2-(1H-imidazol-2-yl)ethyl]-1H-imidazole
3-(2,1,3-benzoxadiazol-5-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-benzyl-3-ethyl-1-(5-fluoro-1H-indole-2-carbonyl)-1,4-diazepan-5-one
methyl 2-{1-[7-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazole-5-carbonyl]-3-oxopiperazin-2-yl}acetate
4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
5-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(5-chloro-2-methoxyphenyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
1-methyl-3-{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}imidazolidine-2,4-dione
3-[1-(3-chlorobenzoyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
4-ethyl-3-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(oxan-2-ylmethoxy)acetamide
[4-benzyl-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]methanol
N-benzyl[(2-methyl-1-benzofuran-7-yl)amino]sulfonamide
2-(2-{1-[2-(1H-indol-1-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-3-(2-methylphenyl)-3-phenylpropanamide
2-{[2-amino-6-(3-chloro-4-methoxyphenyl)pyrimidin-4-yl]amino}ethan-1-ol
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,3-thiazole-4-carboxamide
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
6-(3-chlorobenzoyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
3-[4-phenyl-5-(quinolin-3-yl)-1H-imidazol-1-yl]propan-1-ol
N-[(4-ethylphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylpiperidine-4-carboxamide
1-(diphenylmethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[3-(2-ethylphenoxy)azetidin-1-yl]-4-(piperidine-1-carbonyl)pyridine
N,N-dimethyl-2-[(1S,5R)-6-(4-phenylbutanoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
[(3R,4R)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(thiophen-2-ylformamido)propanamide
3-[4-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
6-[(3-methoxyphenyl)methoxy]-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
2-[1-(cyclopropylmethyl)-4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-yl]ethan-1-ol
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[2-(naphthalen-2-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N2-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-N4,N4-dimethylpyrimidine-2,4-diamine
(3S,4R)-1-(1,3-benzothiazol-2-yl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-ethyl-N-(2-hydroxyethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-[2-(2-{[5-fluoro-4-(methylamino)pyrimidin-2-yl]amino}ethyl)morpholin-4-yl]-2-methyl-2,3-dihydropyridazin-3-one
3-[(2,3-dimethoxyphenyl)methyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide