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4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(propan-2-yl)pyrrolidin-2-one
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](ethyl)(pyridin-2-ylmethyl)amine
N-[1-(2-phenylethyl)piperidin-3-yl]-2-(phenylsulfanyl)acetamide
{3-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-oxopropyl}urea
6-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-[4-(benzenesulfonyl)piperazine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
ethyl 3-(3-phenylpropyl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-3-carboxylate
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(1,2-oxazol-3-ylmethyl)propanamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}ethan-1-one
5-{3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
(4aS,7aR)-1-(1-methyl-1H-imidazole-2-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-1-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
1-[2-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(3-methylphenoxy)piperidine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-phenoxypropan-1-one
3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-6-[2-(thiophen-2-yl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-(3-{[1-(6-chloropyridazin-3-yl)piperidin-4-yl]amino}butyl)phenol
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-N-(3,5-dimethylphenyl)-2-oxoacetamide
3-methyl-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
(4aS,7aR)-N-ethyl-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
2-(4-acetylpiperazin-1-yl)-2-(2,6-dimethoxy-4-methylphenyl)acetic acid
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
6-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octane-8-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(cyclopropylmethyl)-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-propylacetamide
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
2-[(3-hydroxypropyl)(methyl)amino]-2-(2-methoxy-5-methylphenyl)acetic acid
[4-(furan-2-yl)butan-2-yl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-3-methyl-1H-indole-2-carboxamide
3-[(cyclobutylamino)methyl]-1-(cyclohexylmethyl)-3-hydroxypiperidin-2-one
2,8-dimethyl-4-(4-methyl-2-phenylpiperazine-1-carbonyl)quinoline
2-methoxy-1-{1'-[2-(morpholin-2-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(2-{[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl][(2-methylphenyl)methyl]amino}ethyl)dimethylamine
(1R,6S)-6-[3-(2-methyl-1H-indol-1-yl)propanamido]cyclohex-3-ene-1-carboxamide
2-(4-methoxyphenyl)-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[3-(2-ethylphenoxy)azetidine-1-carbonyl]cyclopropane-1-carboxamide
N-cyclopropyl-3-{1-[2-(4-phenylphenyl)acetyl]piperidin-3-yl}propanamide
6-(aminomethyl)-N-[2-(1H-indol-3-yl)ethyl]-2-methylpyrimidin-4-amine
N-[(2,4-dimethoxyphenyl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
[(4aS,8aR)-6-(2-methyl-4-phenylpyrimidine-5-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
methyl[(1-methyl-1H-imidazol-2-yl)methyl]({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)amine
N,N-dimethyl-4-[4-(pyridin-4-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
5-[(2-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}ethyl)sulfanyl]-1H-1,2,3-triazole
1-(3-fluorophenyl)-N-(isoquinolin-5-ylmethyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide