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1,N3-dibenzyl-N5-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-cyclopropyl-N-{2-[methyl(phenyl)amino]propyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-(2-methoxyethyl)-6-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,3-benzoxazole
1-[(4-methyl-1H-imidazol-5-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)oxolane-3-carboxamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
1-(2-fluorophenyl)-N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
{1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
7-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4H-chromen-4-one
1-(4-cyano-2-ethylphenyl)-3-[2-(3,5-dimethoxyphenyl)-2-hydroxyethyl]urea
1-(2-methylfuran-3-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
5-(2,3-dimethoxybenzoyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-(1H-pyrazol-4-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]butan-1-one
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2,2-bis(prop-2-en-1-yl)pyrrolidine
N-[2-(benzylsulfanyl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-[1-(4-methoxybenzoyl)piperidin-3-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-methoxy-2-methyl-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)acetamide
4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
3-(piperidine-1-carbonyl)-2-[4-(propan-2-yloxy)phenyl]pyridine
1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
methyl[1-(pyrazin-2-yl)propan-2-yl](1,3-thiazol-4-ylmethyl)amine
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-benzofuran-2-carboxamide
ethyl 5-(2H-1,3-benzodioxole-5-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-methanesulfonyl-4-(6-methyl-2-propylpyrimidin-4-yl)-1,4-diazepane
2-[5-({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}carbamoyl)pyridin-2-yl]benzoic acid
1-methyl-4-phenyl-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,3S)-3-(2-aminoethoxy)-7-(2-propoxybenzoyl)-7-azaspiro[3.5]nonan-1-ol
1-[1-(2-chlorobenzoyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
9-(2-methoxyethyl)-1-methyl-4-(1H-pyrazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(3-methylthiophen-2-yl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-(dimethylamino)butan-1-one
5-(morpholin-4-ylmethyl)-N-[2-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(4-hydroxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazole-5-carboxamide
(2S)-2-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]-2-phenylacetamide
4-{1-[1-(5-chloropyridin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-(1-{7-[(2,3,6-trifluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-{[(2S,4S)-4-fluoro-1-(1-methylcyclopropanecarbonyl)pyrrolidin-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-sulfonamide
1-(1H-imidazole-5-carbonyl)-3-(thiophene-2-carbonyl)piperidine
3-{1-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
N-[2-(4-fluorophenoxy)pyridin-3-yl]-3-propoxypiperidine-1-carboxamide
3,5,7-trimethyl-N-[(3S)-pyrrolidin-3-yl]-1H-indole-2-carboxamide
{[3-(azocane-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl}diethylamine
N-{[7-(1H-indole-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
(1S,5R)-6-(cyclobutylmethyl)-3-(5-hydroxypyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-acetyl-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}benzene-1-sulfonamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(thiophen-3-ylmethyl)-1,4-diazepan-5-one
1-(morpholin-4-yl)-3-[1-(1-phenylcyclohexanecarbonyl)piperidin-3-yl]propan-1-one