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2-(3-{2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}piperidin-1-yl)acetamide
N-(2-hydroxyethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-[4-(3-phenylbutyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
3-[4-methyl-2-(pyrimidin-5-yl)phenyl]-1,3-oxazolidin-2-one
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(pyridin-3-yl)propan-1-one
2-({1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-imidazole
2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
2-(2-{[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]methyl}phenoxy)acetic acid
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-3-carboxylic acid
N-ethyl-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(2E)-3-phenylprop-2-en-1-yl]butanamide
1-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,6-tetrahydropyridin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(3-cyano-2-methyl-1H-indol-1-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
3-(pyrrolidine-1-carbonyl)-2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine
2-amino-6-(4-hydroxy-3-methoxyphenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(naphthalen-2-yloxy)propanamide
1-cyclohexyl-1-(2-hydroxy-2-phenylethyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
5-methyl-N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
3-{[(2-acetamidoethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(1R,5S,8S)-8-methoxy-N-{4-[2-(pyridin-2-yl)ethoxy]phenyl}-3-azabicyclo[3.2.1]octane-3-carboxamide
4-(1-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl}ethyl)morpholine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-benzyl-N-(cyclobutylmethyl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
N,N-dimethyl-2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
3-fluoro-N-[4-(pyrimidin-5-yl)phenyl]benzamide
1-(1-{6-[(furan-2-ylmethyl)(methyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
1-{2-chloro-4-[2-(furan-2-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,4-triazole
2,6-dimethyl-4-[4-(thian-4-yl)piperazine-1-carbonyl]quinoline
2-methyl-6-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidin-4-ol
N,N-dimethyl-6-[3-(morpholin-4-ylmethyl)phenyl]pyridazin-3-amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-(furan-2-yl)benzamide
N-[4-(azepan-1-yl)butyl]-1H-pyrazole-4-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]-2-(6-methoxypyridin-3-yl)acetic acid
5-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
1-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
3-(3,4-dimethoxyphenyl)-1-{3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]-2-methylpiperidine
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(6-hydroxypyrimidin-4-yl)methyl]propanamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-[(3-fluorophenyl)methyl]-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-2-carboxamide
4-[(3-fluorophenyl)methyl]-1-[3-(1H-indol-3-yl)propanoyl]-1,4-diazepan-5-one
(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-ethyl-3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-4H-1,2,4-triazole