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1-methyl-4-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}ethyl)piperazine
(3S,4R)-4-phenyl-1-(3,3,3-trifluoropropyl)pyrrolidine-3-carboxylic acid
4-({3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
1-[(5-ethylfuran-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperazine-1-sulfonamide
methyl 1-benzyl-3-cyclopropaneamido-5-[(4-hydroxybutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(3R,4R)-1-(1-benzofuran-5-ylmethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)quinoxaline
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)thiophen-2-yl]ethan-1-one
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-methylquinoline
6,6-dimethyl-1-phenyl-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1'-[4-(pyrrolidin-3-yl)benzoyl]spiro[indene-1,4'-piperidine]
3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-ylmethyl}benzonitrile
3-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-[3-(4-hydroxyphenyl)propyl]-2-(propan-2-yloxy)propanamide
1-(azocan-1-yl)-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-[(2S)-2-[3-(2,4-dimethylphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethan-1-one
N-cyclopropyl-3-[1-(2,5-dimethylbenzoyl)piperidin-3-yl]propanamide
(2S)-2-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-phenylacetamide
N-{1-[1-(2-acetamidoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
2-cyclopropanecarbonyl-8-[(4,5-dimethylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N4-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(methylsulfanyl)pyrimidine-4,6-diamine
3-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
9-(3-hydroxy-2-methylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-(4-methoxy-3-pentanamidophenyl)-1,2,3-thiadiazole-4-carboxamide
6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(3-methoxyphenyl)-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
2-(adamantan-1-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
1-(2-chloro-4,6-dimethylphenyl)-3-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}urea
1-[(2,3-difluorophenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(3-methoxyphenyl)methyl]amine
N'1-[(2-methoxyphenyl)methyl]-N'1-(prop-2-en-1-yl)cyclopropane-1,1-dicarboxamide
3-(4-cyclohexanecarbonylpiperazin-1-yl)-N-(thiophen-2-ylmethyl)propanamide
{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-3-ylmethyl)amine
8-(1H-imidazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
2-amino-4-[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-[(3S,4R)-1-[1-(2,3-dimethylphenyl)piperidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-(4-chlorophenyl)-5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-hydroxypiperidin-4-yl}-1-benzofuran-2-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazine
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-ethyl-8-(5-methyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-(cyclohex-1-en-1-yl)acetyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2H-1,3-benzodioxole-5-carboxamide
5-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
7-methoxy-3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one