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2-methoxy-5-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
{1-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-3-propylpiperidin-3-yl}methanol
N-(4-methoxyphenyl)-1-(2-{[2-(trifluoromethyl)phenyl]formamido}ethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 1-[(3S,5S)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
7-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-indole
5-methanesulfonyl-2-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrimidin-4-amine
4-{5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-3-methylpyridine
4-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(2H-1,3-benzodioxol-5-yl)-3-(2-methoxyethyl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-(4-methoxy-2-methylphenyl)-3-(thiophene-2-sulfonamidomethyl)piperidine-1-carboxamide
2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
N-[(2-chlorophenyl)methyl]-3-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}propanamide
1-[1-(3,4-difluorobenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
(4aS,8aR)-1-(3-aminopropyl)-6-(1H-1,3-benzodiazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methylpyrazin-2-yl)methyl]piperidine-3-carboxamide
6-(2,2-dimethylpropyl)-N-[2-(1H-indol-3-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
2-(2-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}ethyl)phenol
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(4-fluorobenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}cyclohexanecarboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
5-ethyl-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
1-ethyl-N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[2-(ethylsulfanyl)phenyl]-3-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}urea
2,5-dimethyl-3-{3-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]phenyl}pyrazine
(1s,4s)-4-{[methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}cyclohexan-1-amine
{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
(3R,5S)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-hydroxy-4-propoxy-5-(1H-pyrazol-4-yl)benzoic acid
N-(1H-imidazol-2-ylmethyl)-4-[(1-methoxypropan-2-yl)sulfamoyl]benzamide
4-phenyl-3-{1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[2-(trifluoromethyl)phenyl]methyl}cyclopropanamine
8-(furan-3-ylmethyl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1H-1,3-benzodiazol-2-yl)-N-(6-methoxy-2H-1,3-benzodioxol-5-yl)pyrrolidine-1-carboxamide
2-[4-(5,6-dimethylpyrimidin-4-yl)-1,4-diazepan-1-yl]-1,3-benzothiazole
4-[4-(3-chlorophenyl)-5-methyl-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
(2S)-1-{4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carbonyl}pyrrolidine-2-carboxamide
2-[8-(1-methoxypropan-2-yl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-(2-{[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
6-chloro-2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(1H-1,2,4-triazol-1-yl)adamantane-1-carboxamide
1-(cyclohexyloxy)-3-[(pyrimidin-2-yl)amino]propan-2-ol
1-[4-(2-ethylphenyl)piperazin-1-yl]-3-methoxy-2,2-dimethylpropan-1-one
7-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-fluorophenyl)-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)morpholine
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
5-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazole