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4-(3-methoxypropyl)-N-(2-phenylphenyl)piperazine-1-carboxamide
1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
5-{[2-(2,3-dihydro-1H-inden-1-yl)acetamido]methyl}thiophene-2-carboxylic acid
N-(cyclopropylmethyl)-4-{[2-(5-methylfuran-2-yl)ethyl]sulfamoyl}benzamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyridine-2-carboxamide
4-[2-(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperazin-1-yl)ethyl]morpholine
3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1-phenylpyrrolidin-2-one
(1R,2R,6S,7S)-4-[(3-methylthiophen-2-yl)sulfonyl]-4-azatricyclo[5.2.1.02,6]decane
4-[(3-methoxyphenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}benzonitrile
2-(2-{[3-(methylsulfanyl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(3S,4S)-1-(4-{[(3-methylthiophen-2-yl)methyl]amino}benzoyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-(2-methylpropyl)pyrimidin-2-amine
1-(2-cycloheptylethyl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
(3R)-1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidin-3-ol
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
1-methyl-6-propyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-ethyl-N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
4,4,4-trifluoro-1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]butan-1-one
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[2-(pyridin-2-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
N'-(3-chloro-4-fluorophenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]butanediamide
methyl (1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
N-(3-hydroxypropyl)-2-(2-methylphenoxy)-N-[(5-methylthiophen-2-yl)methyl]acetamide
6-methyl-2-{[(4-methyl-1,4-oxazepan-6-yl)methyl]amino}pyridine-3-carbonitrile
2-(2,2-dimethylpropanoyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-{2-[3-(3-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-6-(piperidine-1-carbonyl)pyrazine
1-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]-N,N-dimethylbutanamide
1-({5-[1-(cyclopropylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(4-methylpyridine-3-carbonyl)piperidine-4-carboxylic acid
1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-phenyl-1,4-diazepane
N-[(3-chlorophenyl)methyl]-3-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]propanamide
2-(2-methoxyethyl)-8-(4-methyl-1H-imidazole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-methoxy-1-[1'-(3-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(3-methylphenyl)-3-{1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}propanamide
({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-phenyl-1,4-diazepane
(1R,5R)-3-(4-chloro-3-fluorobenzoyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
2-(5-methylpyrazine-2-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
8-(3,5-difluorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4S)-N,N-diethyl-1-(1H-imidazol-2-ylmethyl)-4-(2-methylfuran-3-amido)pyrrolidine-2-carboxamide
N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
N-[2-(4-methoxyphenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
methyl (2S,4S,5R)-5-(2-fluorophenyl)-4-{[(3-methoxyphenyl)methyl]carbamoyl}-1-methylpyrrolidine-2-carboxylate