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N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)furan-2-carboxamide
3-[hydroxy(phenyl)methyl]-4-(4-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,4R)-1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
4-[2-(dimethylamino)ethyl]-11-{[(3-methylphenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-2-[(2-fluorophenyl)methyl]-1,6-dimethyl-1,4-dihydropyridin-4-one
2-{[4-(2-chlorophenyl)-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
6-phenyl-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-(2,5-difluorophenyl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
(1R,5S,8S)-8-methoxy-N-(3,4,5-trimethoxyphenyl)-3-azabicyclo[3.2.1]octane-3-carboxamide
8-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-(7-methoxy-4-methylquinazolin-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}piperidine-4-carboxamide
3-{1-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]azetidin-3-yl}pyridine
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-{[1-(3,4-difluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
8-methoxy-2-(4-methoxy-3-methylphenyl)-5-(quinoxalin-5-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-(4-tert-butylbenzoyl)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidine
3-(naphthalene-2-carbonyl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
6-(4H-1,2,4-triazol-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}pyridine-2-carboxamide
1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
1-(3-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)azepan-2-one
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)-N-propylacetamide
N-(adamantan-1-yl)-2-chloro-5-acetamidobenzamide
N-cyclopropyl-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2-hydroxypropyl)-N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
6-chloro-2-{2-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
3-[(2R,3R,6R)-5-[2-(methylamino)pyridine-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[(2-methylphenyl)methyl]-N-(2-methylpropyl)acetamide
N-cyclopropyl-3-(1-methyl-1H-pyrazol-5-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
(3R,5S)-5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-3-amine
N-{3-oxo-3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}acetamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)methylamine
3-(diphenylmethyl)-5-(2-ethoxyethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
6-{[2-(3-methoxypropyl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzothiazol-2-one
(2S)-2-[5-oxo-3-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
4-(3,4-dimethoxyphenyl)-3-(4-hydroxy-3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(hydroxymethyl)-1-(2-phenylquinolin-4-yl)piperidin-3-ol
6-[(3,5-dimethoxyphenyl)methoxy]-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-(propan-2-yl)-1,4-diazepan-2-one
N-[3-(dimethylamino)propyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(2-ethoxypyridin-3-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
9-(3-methoxybenzenesulfonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-[2-(propan-2-yloxy)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(3-fluorophenyl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazin-2-one
2-[3-(1H-imidazol-1-yl)propyl]-9-(3-methyl-1H-pyrazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-(propan-2-yl)-1H-pyrazole
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-methoxy-4H-pyran-4-one