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N-[(5-fluoro-2-methylphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,9aR)-3-benzyl-2-methyl-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]benzoic acid
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
4-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-1,4-diazepane-1-carbaldehyde
2-(2-{[(dimethylcarbamoyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)acetic acid
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-{[(5-cyanopyridin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methoxypyridazine
ethyl 1-{[5-(2,5-dimethoxyphenyl)-2-hydroxyphenyl]methyl}piperidine-2-carboxylate
1-methyl-5-(2,3,4-trimethoxyphenyl)-1H-1,2,3,4-tetrazole
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-4-fluorobenzamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxyacetamide
1-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}azepan-2-one
4-(4,6-dimethylpyrimidin-2-yl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(3S,4R)-4-(hydroxymethyl)-1-(5-phenoxyfuran-2-carbonyl)piperidin-3-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]acetamide
4-(5-ethylfuran-2-yl)-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-1,2,3-triazole
N-[2-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(2-methylphenyl)-3-phenylpropanamide
4-[5-cyclobutyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
3-fluoro-N-({7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
methyl 3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}amino)-4-methoxybenzoate
5-ethyl-N,2,3-trimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-methyl-5-[(2S)-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl]-1,2,4-oxadiazole
4-(4-{[(2-methoxyethyl)amino]methyl}phenyl)phenol
7-(1-benzothiophen-3-yl)-4-(pyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-fluorophenyl)-5-(thian-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1,3-thiazole-4-carboxamide
5-{[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]methyl}thiophene-2-carboxylic acid
1-(5-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
3-{1-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperidin-3-yl}propanamide
(4aS,7aR)-1-(2,4-dimethylbenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-6-{4-[1-(propan-2-yl)piperidine-3-carbonyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
2-[(1-benzyl-4-phenylpiperidin-4-yl)formamido]-N-methylacetamide
3-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
4-(4-chlorophenyl)-1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-4-ol
2-({[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl)amino)-N,N-dimethylpropanamide
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-2-methoxy-N-(2-methoxyethyl)acetamide
N-(1-methoxybutan-2-yl)-3-[(oxan-4-yl)sulfamoyl]benzamide
[3,3-dimethyl-1-(pyridin-3-yl)butyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(4-fluorophenyl)ethyl]-N-methylacetamide
4-{1-[6-(pyridin-4-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
(3R,4S)-1-cyclobutanecarbonyl-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
1-methyl-2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-1,3-benzodiazole
3-(2H-1,3-benzodioxol-5-yl)-N-{[5-chloro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-methoxy-N-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
[(3R,4R)-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol