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3-({1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-yl}methyl)benzoic acid
3-{5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-[(5-methylthiophen-2-yl)sulfonyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
N-(5-methyl-1H-pyrazol-3-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
2-{[4-(1-phenylethyl)-5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-[(2,5-difluorophenyl)methyl]-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{5-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]oxolane-2-carboxamide
1-methyl-3-(5-phenyl-1,3,4-thiadiazol-2-yl)-1-(thiophen-3-ylmethyl)urea
1-[3-(4-fluorophenyl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
(1R,7S)-3-(4-fluoro-2-methylphenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-2-(thiophen-2-yl)pyrimidin-4-ol
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1,4-dimethylpiperazin-2-yl)acetamide
N-methyl-4-(1H-pyrazol-3-yl)-N-[1-(pyrimidin-4-yl)ethyl]benzamide
2-methyl-5-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazine
3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2,5-dioxoimidazolidin-1-yl)-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}acetamide
3-chloro-4-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenol
N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
3-(1-methylpiperidin-3-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
(3R,4R)-4-(azepan-1-yl)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-ol
N-(1-{[(2,3-dihydro-1H-inden-1-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-fluoro-2-{3-[(4-methylpiperazin-1-yl)methyl]piperidine-1-carbonyl}phenol
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-3-carboxamide
N-{3-[cyclopentyl(methyl)amino]propyl}-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
6-methoxy-3-methyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1-benzofuran-2-carboxamide
(5-{4-[2-(morpholin-4-yl)ethyl]piperazine-1-carbonyl}-1H-1,3-benzodiazol-2-yl)methanol
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
5-(3,3-dimethylbutyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2-hydroxypropyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
(cyclopropylmethyl)(2-methoxyethyl)[(4-methylphenyl)methyl]amine
9-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-{[2-(furan-2-yl)phenyl]methyl}-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(5-methylthiophen-2-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
ethyl 4-[3-(2-{[(2-chlorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]piperidine-1-carboxylate
[(2S,6S)-4-[(4-fluoro-3-methoxyphenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-cycloheptyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-1,2-dihydrophthalazin-1-one
2-[2-(1H-imidazol-1-yl)ethyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-1-carboxamide
methyl 3-{[(3-ethyl-1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-(2-fluorobenzamido)benzoate
2-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-4-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
8-(2-methoxybutanoyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(3S,9aR)-3-benzyl-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 6-(3-fluorobenzoyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate