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2-(4-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperazin-1-yl)pyrimidine
2-(2-fluorophenyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
2-(ethylsulfanyl)-5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
8-(2-aminopyridine-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]butanamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(quinolin-5-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
5-cyclopropanecarbonyl-1'-[(2S)-1-(propan-2-yl)pyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methoxy-N-({5-[(4-methoxy-2,3-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
(4aR,7aS)-N,N-dimethyl-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-cyclohexyl-4-{3-[(2-methylpyrrolidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}piperazine
N-[furan-2-yl(phenyl)methyl]-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
methyl 3-{[5-(1,3-benzothiazol-2-ylmethyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-[4-(morpholin-4-yl)phenyl]pyridine-3-carbonitrile
2-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(pyrazin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]-4-aminopyrimidine-5-carbonitrile
4-{4-[(2,3-dimethoxyphenyl)methyl]piperazin-1-yl}butan-1-ol
4-benzyl-1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-{4-[4-(azepane-1-carbonyl)-7,8-dimethylquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
N-ethyl-3-(1H-imidazol-2-yl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
2-[(3-methylpyrazin-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-3-tert-butyl-1,2,4-oxadiazole
3-[(3R,4S)-1-[2-(3,4-dimethylphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-acetamido-N-[2-(3-phenylpropoxy)phenyl]propanamide
1-cycloheptyl-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]azepan-4-ol
1-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-(2,3-dichlorophenyl)-1-[(2S)-oxolan-2-ylmethyl]-1H-1,2,3-triazole
N-{2-[(2-fluoro-4-methoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
1-(pentan-3-yl)-4-[(1E)-1-phenylprop-1-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-[3-(pyridin-4-yl)azetidin-1-yl]pyrimidine-2,4-diamine
(1R,5S)-6-[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-6-azabicyclo[3.2.1]octane
4-[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]-1-oxaspiro[4.4]nonan-2-one
4-({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
N-({1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-[2-(5-methylfuran-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
3-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
N-[(2R,3R)-1'-[(3,4-dimethylphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
ethyl 2-{methyl[5-({[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)pyrimidin-2-yl]amino}acetate
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
(1S,5R)-6-(1H-indole-6-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
1-methyl-3-(3-{4-[(1-methyl-1H-pyrazol-4-yl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide