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4-cyano-N-[3-(2-methoxyethoxy)phenyl]-4-phenylpiperidine-1-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
4-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}-N,N-dimethylbutanamide
1-(propan-2-yl)-4-{1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}piperidine
1-(3,5-dimethylphenyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
(3aS,7aR)-2-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{1-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
ethyl 1-[(4-methoxyphenyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
1-[3-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]ethan-1-one
[(1-cyclopentylpiperidin-4-yl)methyl][(2-methylphenyl)methyl](oxolan-2-ylmethyl)amine
2-methoxy-N-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[(1-hydroxycyclohexyl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
N-({1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
N-[3-chloro-4-(propylcarbamoyl)phenyl]-3-(pyridin-2-yl)azetidine-1-carboxamide
4-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
N-[3-(methylsulfanyl)phenyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(4-methylpiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N,2-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1-benzofuran-5-carboxamide
4-(1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,2,5-thiadiazole-3-carboxamide
1-(6-cyanopyridin-2-yl)-4-(4-fluorophenoxy)piperidine-4-carboxylic acid
8-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R)-3,4,4-trimethyl-1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)oxolane-3-carboxamide
1-[4-(pyridin-2-ylmethoxy)phenyl]-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
2-methyl-4-{pyrazolo[1,5-a]pyridin-7-yl}-5H,6H,7H-cyclopenta[d]pyrimidine
5-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
4-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-6-methoxypyrimidin-2-amine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
1-{4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-methyl-2-[3-(3-methylthiophen-2-yl)benzoyl]-1H-imidazole
2-(azepan-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(2H-1,3-benzodioxol-5-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1,2,4-triazin-3-amine
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-(cyclohexylmethyl)piperazin-2-yl}ethan-1-ol
4-methoxy-N-({6-methyl-2-[methyl(1H-pyrazol-5-ylmethyl)amino]quinolin-3-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyridin-4-yl)acetamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-4-[(4-methylphenyl)methyl]piperazin-2-one
4-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-1-phenylpiperazin-2-one
N-[(4-ethylphenyl)methyl]-5-(3-fluorophenyl)-N-methyl-1,2,4-triazin-3-amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
1-(furan-3-ylmethyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
2-amino-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
N-(2-methylprop-2-en-1-yl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
[5-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)furan-2-yl]methanol