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[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(4-methanesulfonylphenyl)methyl]methylamine
4-(1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-1H-1,2,3-triazol-4-yl)quinoline
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
2-cyclopropyl-9-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-methyl-N-[(4-phenoxyphenyl)methyl]benzamide
4-(cyclopropylmethyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
4-acetyl-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
N,N-dimethyl-1-({2-[(4-methylphenyl)methoxy]phenyl}methyl)azepan-4-amine
N-methyl-4-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]benzamide
2-oxo-2-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]acetamide
8-chloro-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)quinoline-2-carboxamide
3-[(1-acetylpiperidin-3-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(propan-2-yl)amino]pyridine-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(2-methoxyphenyl)benzamide
4-{[5-(2,4-dimethoxy-3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrimidine
N-[3-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-oxopropyl]methanesulfonamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylquinoxaline-6-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidine-3-carbonitrile
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-2-ethylpyrimidine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-5-fluoropyridine-3-carboxamide
1-{3-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]propyl}pyrrolidin-2-one
1-(1-carbamoylpiperidine-3-carbonyl)-4-phenylpiperidine-4-carboxylic acid
5-methanesulfonyl-4-(piperidin-3-yl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidin-2-amine
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(naphthalen-2-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
7-benzyl-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(3aR,6aS)-1-oxo-5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-(3-methylbutanoyl)-4-[2-(1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-4-ylsulfanyl)acetamide
2-(4-methoxyphenyl)-N-[4-(4-{[(4-methyl-1,3-thiazol-2-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(2-phenoxyethyl)piperidine-3-carboxamide
2-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}urea
4-[1-(3,3,3-trifluoro-2-methylpropyl)piperidin-4-yl]pyrimidine
N-butyl-N,5-dimethyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-amino-6-(2,2-dimethyloxan-4-yl)-5-methyl-4-(piperidin-4-yl)pyridine-3-carbonitrile
4-benzyl-1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
1-(2,4,6-trimethyl-3-{1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-(trifluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[(6-chloropyridin-3-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-methoxypropan-1-one
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2,4-difluorophenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-ethyl-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-{[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}ethan-1-ol
N-(2-methoxyphenyl)-3-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}propanamide
N-ethyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-4-ylmethyl)acetamide
N,N-dimethyl-5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
4-{2-methyl-2-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]propyl}morpholine