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9-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-3,9-diazaspiro[5.6]dodecane
3-(2,5-dimethylpyrimidin-4-yl)-2-methoxyquinoline
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1H-pyrrole-3-carbonitrile
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)pyrrolidin-2-one
N-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
6-(2-aminoethyl)-N-[(5-chloro-1-benzothiophen-3-yl)methyl]-2-methylpyrimidin-4-amine
1-[(4-fluorophenyl)methyl]-5-(3-methylpyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-{[(2R)-1-hydroxybutan-2-yl]amino}-N-[(3S)-2-oxoazepan-3-yl]pyridine-2-carboxamide
5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-2-(propan-2-yl)-1,3-benzoxazole
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
[(4-cyclopropyl-5-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
[3-(2-phenylethyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl]methanol
N'-(2,5-dimethoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanediamide
N-phenyl-4-[4-(1H-pyrazol-4-yl)butanamido]piperidine-1-carboxamide
methyl 4-({[2-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-oxopyrrolidin-2-yl)ethyl]amino}methyl)benzoate
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
7-chloro-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-N-(oxolan-2-ylmethyl)quinazolin-4-amine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-(aminomethyl)-4-[(1R)-1-(4-chlorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-4-({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}amino)piperidine-1-carboxamide
2-[5-cyclopropyl-4-(3-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-4-phenylazepane-1-carboxamide
6-ethyl-2-methyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide
2-(4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)phenol
methyl 5-[(cyclohexylmethyl)carbamoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
(2S)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-({[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[3-(1,2-oxazinan-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(2-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
2-(cyclopent-2-en-1-yl)-1-{4-[(3-methoxypropyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
N,N-diethyl-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}ethan-1-one
(2S,4R)-4-amino-1-[2-(methylsulfanyl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N'-cyclopentyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methylbutanediamide
N-[1-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]furan-2-carboxamide
4-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)thiomorpholine
7,7-dimethyl-2-[1-(phenoxymethyl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-[2-(dimethylamino)ethyl]-N-[3-(2-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(4-methyl-1H-imidazole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one