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2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N-(4-fluoro-2-methylphenyl)acetamide
(9aR)-8-(cyclohexylmethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-benzyl-3-(2-methoxyethyl)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)acetamide
5-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}pyrimidin-2-amine
3-[1-(pyridin-3-yl)propan-2-yl]-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)azocane
{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}(methyl)(piperidin-3-ylmethyl)amine
N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
2-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
4-[7-(1-phenylcyclopropaneamido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]pyridin-1-ium-1-olate
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N'-[2-(1H-indol-1-yl)ethyl]-N'-methyl-N-(5-methyl-1,2-oxazol-3-yl)ethanediamide
1-(cyclopropylmethyl)-N-ethyl-5-[2-(pyridin-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 5-{[(2,6-difluorophenyl)methyl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-(diphenylmethyl)-N-(1-phenylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-pentyl-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[3-(pyrrolidin-1-yl)butyl]acetamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[3-(dimethylamino)pyrazin-2-yl]pyrrolidin-3-yl]methanol
1-[3-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)propyl]piperidin-3-ol
N-(2-hydroxyethyl)-4-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}pyridine-2-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
1-(benzenesulfonyl)-4-(1,2-oxazole-5-carbonyl)piperazine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-phenylacetamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-[(3R,4S)-1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-{1-[4-(2-ethoxypyridin-3-yl)phenyl]ethyl}acetamide
1-{4-[2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-7-yl]piperidin-1-yl}-2-methylpropan-1-one
1-methyl-4-(4-methyl-1H-pyrrole-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(3-fluorophenyl)-3-{1-[1-(2-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-[1-(methoxymethyl)cyclopropyl]-3-methyl-1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
1-{4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}ethan-1-one
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
3-{3-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2H-chromen-2-one
3-cyclohexyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-methyl-5-oxo-N-[2-(piperidin-1-ylmethyl)phenyl]-1,4-diazepane-1-carboxamide
(furan-2-ylmethyl)({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})(prop-2-en-1-yl)amine
3-(1-cyclobutylpiperidin-4-yl)-N-cyclopropylpropanamide
4-(3-aminopiperidine-1-carbonyl)-6-ethyl-1,2-dihydropyridin-2-one
N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-methyl-2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-1,3-benzodiazole
N-(2-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-ethyl-3-(piperidine-1-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-ethyl-4-[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-2-one