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4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]thiomorpholine
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
3-butyl-1-(1-cycloheptyl-5-oxopyrrolidin-3-yl)urea
7-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1-benzofuran-2-carboxamide
8-(3-fluorobenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-(3-phenylpropyl)piperidin-2-one
ethyl 1-{[4-(methylsulfanyl)phenyl]carbamoyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
methyl 9-(cyclopentyloxy)-3-(6-methylpyridine-3-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(4-chlorophenyl)-N-[1-(cyclopropylmethyl)azepan-3-yl]-4-methyl-1H-pyrazole-3-carboxamide
8-[2-(4H-1,2,4-triazol-4-yl)ethyl]-8-azaspiro[4.5]decane-7,9-dione
2-(2-{[2-(trifluoromethyl)pyrimidin-4-yl]amino}ethoxy)ethan-1-ol
(1S,5R)-6-(cyclopropylmethyl)-3-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-1-(5-fluoropyridin-3-yl)urea
5-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
8-(2-cyclopropylpyrimidine-5-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1,6-dimethyl-4-oxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,4-dihydroquinoline-3-carboxamide
8-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
3-(3-cyanopiperidine-1-carbonyl)-N-(oxan-4-yl)benzene-1-sulfonamide
2-acetamido-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
N'-cyclopentyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanediamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(2-hydroxyphenoxy)ethan-1-one
2-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-4-methyl-1H-imidazole
2-[4-(ethanesulfonyl)piperazin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
2-ethyl-8-(2-{methyl[(4-methylphenyl)methyl]amino}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
5,8-dimethyl-2-{[(1,3-thiazol-2-ylmethyl)amino]methyl}quinolin-4-ol
N-methyl-4-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carbonyl]morpholine-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(dimethylamino)-2-(4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
4-ethyl-1-[(3-fluorophenyl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amine
2-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(cyclopropylmethyl)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidine-3-carboxylic acid
3-(2-aminoethyl)-4-(3-phenoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(2S,6S)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(3-fluorophenyl)ethyl]propanamide
(4S,6R)-N-[3-(2-methoxybenzamido)phenyl]-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
2-{3-[(3-methyl-3-phenylpiperidin-1-yl)methyl]phenoxy}acetamide
1-[1-(3-acetyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
2-(2-chlorophenyl)-N-[2-(dimethylamino)ethyl]-N,3-dimethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-(2-methanesulfonylethyl)urea
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-[(2-methylpropyl)amino]-N-(propan-2-yl)pyrrolidine-2-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-(pyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methoxy-3-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-indazole
(1R,5R)-3-methanesulfonyl-6-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-(piperazin-1-yl)-2-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydropyridazin-3-one