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4-(4-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
ethyl 4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]thiolan-3-amine
2-butyl-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[2-(pyridin-2-ylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3aR,6aR)-2-[2-(2-methoxyphenyl)acetyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-N-(2-phenylethyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,3R)-3-amino-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]cyclopentane-1-carboxamide
1-[(4-methoxyphenyl)methyl]-4-(5-methoxypyrimidin-2-yl)piperazin-2-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
(1,4-dioxan-2-ylmethyl)(methyl){[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(thiophen-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
({4-ethyl-5-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1-(propan-2-yl)piperidine-4-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(3,4-difluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]butan-1-one
1-(adamantan-2-yl)-3-(pyrrolidin-1-yl)piperidine
2-(2,3,4-trifluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
6-(cyclopropylmethoxy)-4-(3-fluorobenzoyl)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)cyclopropanesulfonamide
3-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-1-(2-methoxyphenyl)urea
methyl (1R,5S,6R)-6-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-3-yl)methanamine
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-cyclohexyl-2-(4,5-dimethyl-2-oxo-2,3-dihydro-1,3-oxazol-3-yl)butanamide
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2,5-dimethylfuran-3-carboxamide
2-{[2-amino-6-(2-chloro-4-fluorophenyl)pyrimidin-4-yl]amino}ethan-1-ol
2-{2-[4-(4-methoxyphenyl)-3,3-dimethyl-5-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
methyl 1-[(3R,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]pyridin-4-amine
2-methoxy-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
ethyl 1-(2,6-dimethylpyrimidine-4-carbonyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-[(3R,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(3-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methanol
1-{5-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
{1-[2-(1H-imidazol-1-yl)ethyl]-3-propylpiperidin-3-yl}methanol
2-(adamantan-1-yl)-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]acetamide
{3-[(4-fluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
2-cyclopentyl-N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
3-(4-hydroxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]-2-(thiophen-2-yl)ethan-1-one
3-ethyl-8-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,3S)-3-ethoxy-7-(2-hydroxypyridine-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol