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N-benzyl-4-(pyridin-4-yloxy)piperidine-1-sulfonamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-[(3-phenoxyphenyl)methyl]pyrrolidine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
1-(6-cyclopropylpyrimidin-4-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
1-[1-(2,5-dimethoxybenzenesulfonyl)piperidin-3-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(dimethylamino)-N-{[4-(dimethylamino)-1-ethylpiperidin-4-yl]methyl}-2-(4-fluorophenyl)acetamide
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2-propylpyrrolidine
5-[2-(adamantan-1-yl)acetyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4S,4aS,8aS)-4-phenyl-1-(5-propyl-1,2-oxazole-3-carbonyl)-decahydroquinolin-4-ol
1-(1H-imidazol-4-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[2-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)ethyl]-1H-imidazole
9-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-6-oxa-9-azaspiro[4.5]decane
1-[(4-chloro-3-fluorophenyl)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-{1-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
ethyl 1-(pyridin-4-ylmethyl)-5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-4-ethoxypyrimidine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}propanamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[3-(methylsulfanyl)phenyl]methyl}amine
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-(pyridine-2-carbonyl)-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[3-(phenylsulfanyl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{1-[2-(dimethylamino)ethyl]-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl}-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
ethyl 5-{[2-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-5-oxopyrrolidin-1-yl]methyl}furan-2-carboxylate
1-(3-{4-[(furan-2-ylmethyl)(methyl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
(4aR,7aS)-1-{2-[methyl(1,2-oxazol-3-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[4-(3-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}pyridine-3-carboxylic acid
ethyl 1-{[4-(methoxycarbonyl)phenyl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
ethyl 5-[3-(1H-indol-3-yl)propanoyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}propanamide
8-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
4-[(4aS,8aR)-decahydroisoquinolin-2-yl]-N-[2-(morpholin-4-yl)ethyl]pyridine-2-carboxamide
2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-methyl-3-propyl-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1H-pyrazole-5-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-(1-{1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-4-yl}ethyl)morpholine
2-butyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1,3-benzoxazole-5-carboxamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[2-(pyrazin-2-yl)ethyl]benzamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-propylpyrimidin-2-amine
1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methylpropanamide
methyl (2S,4R)-1-methyl-4-(4-oxo-3,4-dihydroquinazoline-2-amido)pyrrolidine-2-carboxylate