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2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-4-(pyridin-3-yl)pyrimidine
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-{[(3,4,5-trimethoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-[3-methyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]urea
1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,4-diazepan-5-one
N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}azocane-1-carboxamide
1-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-butyl-4-[2-(4-hydroxypiperidin-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
2-(2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(5-chlorothiophen-2-yl)methyl]-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
1-[2-(3-methyl-1H-pyrazol-5-yl)pyrimidin-4-yl]pyrrolidin-3-ol
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
8-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-pyrazol-5-amine
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-(pyridin-2-yl)acetamide
(2E)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazole
5-chloro-3-[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3,3-dimethyl-1-(2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)urea
methyl 5-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1H-1,3-benzodiazol-2-yl)methanol
1-[(3R)-3-hydroxypyrrolidin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
3-(3-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-pyrazole-4-carboxamide
4-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-6-methylquinoline
4-({[2-(1H-imidazol-1-yl)-1-phenylethyl]amino}methyl)-2,6-dimethylphenyl acetate
N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide
1-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-propylpiperazine
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
3-(2-hydroxyphenyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-(2-phenyl-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
1-(4-{[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}phenyl)ethan-1-one
[(6-methoxypyridin-3-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
5-methoxy-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-4-oxo-1,4-dihydropyridine-2-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-({4-[(2,4-dichlorophenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}methyl)-N-methylmethanesulfonamide
(1S,5R)-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1,2,5-oxadiazole-3-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(oxolan-3-yl)benzamide
2-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
4-[7-(1H-imidazol-1-yl)-2,3-dihydro-1,4-benzodioxin-6-yl]-4H-1,2,4-triazole
(3R,4R)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-cyclopropyl-3-methylpiperidin-4-ol
N-[(3-chlorophenyl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
3-[5-(2-aminoethyl)-2-methoxyphenyl]benzonitrile
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(1,3-thiazol-2-ylmethyl)amine
N-[(2-phenoxypyridin-3-yl)methyl]-1-phenylmethanesulfonamide
(4aR,7aS)-N,N-dimethyl-4-[2-(methylamino)pyrimidine-5-carbonyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-(cyclohexylmethyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-6-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide