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5-{2-[(2-methoxyethyl)amino]ethyl}-1-(3-phenylpropyl)pyrrolidin-2-one
2-methoxy-N-[(5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]acetamide
1-ethyl-4-(3-fluoro-2,4-dimethylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S)-2-amino-3-cyclohexyl-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]propanamide
N-[(3S,4R)-1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)(oxan-4-ylmethyl)amine
2-[hydroxy(pyridin-3-yl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(4-methoxybenzamido)-7-oxo-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-[(2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
methyl 3-(cyclobutylmethoxy)-5-(4-methyl-3-oxopiperazine-1-carbonyl)benzoate
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N,N-dimethylbenzamide
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}urea
13-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-methyl-1-(2-phenylethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-(2-fluorophenyl)-5-{imidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-[1'-(2-ethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2,3,5-trimethyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-[1-(4-fluorophenyl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[1-(2,1,3-benzoxadiazole-4-sulfonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
(3S,4S)-4-cyclopropyl-1-(4-ethyl-5-methylpyrimidin-2-yl)pyrrolidine-3-carboxylic acid
5-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
3-[6-amino-5-cyano-4-(5-methoxy-1H-indazol-3-yl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
[(3R,4R)-1-[3-(difluoromethoxy)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-ethyl-2-(4-{[2-(furan-2-yl)phenyl]methyl}piperazin-1-yl)acetamide
5-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
1-(4-methoxyphenyl)-6,6-dimethyl-4-(2,4,5-trifluorobenzoyl)piperazin-2-one
N-(1-benzothiophen-2-ylmethyl)-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N2-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
(3S,4R)-1-[2-(2-ethoxyphenyl)acetyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-(3-methoxyphenyl)-1-(2-methyl-1-benzofuran-7-carbonyl)pyrrolidine
3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
N-benzyl-3-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]-N-methylpropanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
N,3,6-trimethyl-N-(1H-pyrazol-5-ylmethyl)-1-benzofuran-2-carboxamide
(3aS,6aS)-2-[2-(2-chloro-4-fluorophenyl)acetyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3,4-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
4-(4-methoxyphenyl)-3-(1H-pyrazol-5-yl)-4H-1,2,4-triazole
1-cyclohexyl-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[3-(1H-imidazol-1-yl)propyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
[(3-chloro-4-methoxyphenyl)methyl][(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
N-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carboxamide
N-(3,5-dimethoxyphenyl)-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}propanamide
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 5-(2-methyloxane-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
8-(8-chloroquinoline-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine