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N-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N,3-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-methyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
8-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1-oxa-8-azaspiro[4.5]decane
N-cyclopentyl-3-fluoro-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-(thian-4-yl)propanamide
(3aR,6aR)-N-(1H-imidazol-2-ylmethyl)-2-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(3S,4R)-1-(2-fluoro-5-methylbenzenesulfonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-acetyl-N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1H-pyrazole-5-carboxamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-[2-methyl-1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]pyridine-2-carboxamide
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-hydroxy-4-methylpentan-1-one
N-cyclopropyl-1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidine-4-carboxamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-(4,4,4-trifluorobutyl)pyrrolidin-3-ol
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-[3-(3-fluorophenoxymethyl)-5-[(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
(2R,3R,6R)-5-(6-ethylpyrimidin-4-yl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[4-(1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-1,2,3-triazol-4-yl)phenyl]acetamide
N-(1-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
(1S,5R)-6-(4-methyl-1,3-thiazole-5-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrrolidine-2-carboxamide
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
4-[5-(2-chlorophenyl)furan-2-carbonyl]thiomorpholine
4-(3-methylphenoxy)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
N-({7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
2-(dimethylamino)-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
1-(2-methoxyphenyl)-4-[1-(3-phenylpropyl)piperidin-3-yl]piperazine
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(1-phenylbutyl)propanamide
5-ethyl-2-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyridine
1-(5-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
{[1-(piperidin-1-yl)cyclohexyl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-[benzyl(methyl)amino]-3-{4-[(butylamino)methyl]phenoxy}propan-2-ol
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-1-methyl-1H-imidazole-2-carboxamide
N-cyclohexyl-N-methyl-2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pent-2-yn-1-yl)piperidine
3-[(2,4-difluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-cyclopentyl-2-methyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1,3-thiazole-4-carboxamide
4-[3-(4-hydroxyphenyl)propanoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,2-dimethylpiperazine
3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]propanamide
3,5-dimethoxy-N-({1-[2-(methylsulfanyl)acetyl]piperidin-3-yl}methyl)benzamide
6-methyl-3-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one