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N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-(4-methylphenyl)quinoline-4-carboxamide
N-methyl-3-phenyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[4-(methylamino)pyrimidin-2-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(propan-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(1H-imidazol-1-ylmethyl)furan-2-carboxamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(methylsulfanyl)propanamide
5-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-2-methylquinoline
(4aR,7aS)-1-(furan-2-carbonyl)-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]-3,9-diazaspiro[5.5]undecane-2,4-dione
1-phenyl-2-{[4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethan-1-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-[1-(2-cyclohexylethyl)-1H-1,2,3-triazol-4-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
(3S,5S)-5-(cyclopropylcarbamoyl)-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperidine-3-carboxylic acid
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
1-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
7-fluoro-1-(2-methoxyethyl)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1,2-dihydroquinolin-2-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
2-(dimethylamino)-2-(2-methylphenyl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-ethyl-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)butanamide
7-(2-methoxyphenyl)-2-(piperazine-1-carbonyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
3-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
1-(3-methylbutyl)-3-(propan-2-yl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
2-methyl-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-imidazole
N-{1-[(2-methylphenyl)methyl]cyclopropyl}-2-(piperidin-4-yl)acetamide
N-[4-(6-chloro-2H-1,3-benzodioxol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]propanamide
8-[5-(2-chlorophenyl)furan-2-carbonyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4-(hydroxymethyl)-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}piperidin-4-ol
4-(1-{[(2,5-dimethylphenyl)methyl]amino}ethyl)hepta-1,6-dien-4-ol
2-{[2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
3-[(4-methoxyphenyl)methyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[(2,3-difluorophenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[4-(4-hydroxybutyl)piperazin-1-yl]-2-(naphthalen-2-yl)acetic acid
2-(2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-4-(thiophen-2-yl)phenoxy)-1-(4-phenylpiperazin-1-yl)ethan-1-one
3-[(3R,4S)-1-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2,3-dimethoxy-N-(2-methoxyethyl)benzamide
4-[(1-{[1-(3-methylpyrazin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
N,5-dimethyl-N-(oxolan-3-yl)-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(3,6-dimethylpyrazin-2-yl)piperidine-4-carboxylic acid
N-cyclopropyl-N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)cyclohexanecarboxamide
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{2-[1-(2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-fluorophenyl)-3-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea