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1-(2-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
methyl 6-[(2-ethylpiperidin-1-yl)methyl]-3-(furan-2-amido)thieno[2,3-b]pyridine-2-carboxylate
N-methyl-N-propyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-6-methylphenol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(thiophen-2-yl)ethyl]acetamide
N-benzyl{[2-(1H-pyrazol-1-yl)phenyl]amino}sulfonamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(methylamino)methyl]piperidin-2-one
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-(pyridin-4-yl)propanamide
(1S,5R)-3-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-(pentan-2-yl)piperidin-4-amine
4-(4-methyl-1,3-thiazole-5-carbonyl)-2-(4-methylpentyl)morpholine
(3S,4R)-1-[(4-methanesulfonylphenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[1-(4-methanesulfonylphenyl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-[2-(diethylamino)ethyl]-2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-[(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)methyl]-4-(propan-2-yl)morpholine
N-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]methyl}thiophene-2-carboxamide
N-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
4-(2-fluorophenoxy)-1-(2-hydroxyacetyl)piperidine-4-carboxylic acid
2-amino-2-methyl-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
N-ethyl-1-(5-methoxy-1H-indole-2-carbonyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-[2-(dimethylamino)ethyl]-9-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-[(3R,5S)-5-(azepane-1-carbonyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-{[4-(2-phenylethoxy)phenyl]methyl}-2-(trifluoromethyl)morpholine
2-(cyclopropylamino)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)acetamide
ethyl (4aS,8aR)-6-(1-benzoxepine-4-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylate
1-(6-cyclopropylpyrimidin-4-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carboxamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[3-(pyridin-4-yl)propyl]propanamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[4-(1H-pyrazol-1-yl)butan-2-yl]piperazine
(2R)-2-{[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}-3-phenylpropan-1-ol
[(3R,4R)-4-[(dimethylamino)methyl]-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
4-methyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}-1,2,5-oxadiazole-3-carboxamide
N-[(2-methoxyphenyl)methyl]-N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
4-methoxy-N,3-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]benzamide
1-cyclohexanecarbonyl-4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-propyl-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[1-({1-[1-(trifluoromethyl)cyclopropanecarbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-ol
4-[5-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]benzamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(quinoxalin-2-yl)pyrrolidin-3-amine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}acetamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
3-[4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazol-1-yl]propanoic acid
N-[2-(2-methoxyphenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[3-(2-benzyl-5-oxopyrrolidin-2-yl)propanoyl]-1-phenylpiperazin-2-one
3-[2-(2,6-difluorophenyl)ethyl]-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidine
1-(adamantane-1-carbonyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-(3-methoxyphenyl)-1-(oxane-4-carbonyl)piperidine
9-[2-(methylamino)pyrimidine-5-carbonyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one