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4-[1-(3-phenylpropyl)piperidin-3-yl]morpholine
1-ethyl-3-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}piperidine
3-methyl-1-(pyrimidin-2-ylmethyl)-1,2-dihydroquinoxalin-2-one
7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(morpholin-4-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[3-(4-{[2-(cyclohex-1-en-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
(2R,3S,6R)-5-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
N-(2-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
9-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
ethyl 1-{3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidine-3-carboxylate
7,7-dimethyl-2-(morpholin-4-yl)-N-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydroquinazolin-5-amine
{1-[(2-ethylphenyl)methyl]-3-(3-methoxypropyl)piperidin-3-yl}methanol
7-chloro-N-(1-methoxypropan-2-yl)-3,5-dimethyl-1-benzofuran-2-carboxamide
3-amino-N-(3-cyano-4-ethoxyphenyl)pyrrolidine-1-carboxamide
2-methoxy-2-phenyl-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
5-methyl-3-(morpholin-2-ylmethyl)-3,4-dihydroquinazolin-4-one
5-chloro-N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]thiophene-2-sulfonamide
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate
2-{1-[(5-ethylfuran-2-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
1-[2-(4-chlorophenyl)acetyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N5-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N6-(3-methoxypropyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-(2-methylquinolin-5-yl)urea
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}[1-(furan-2-yl)ethyl]amine
2-(1H-indazol-1-yl)-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-[(prop-2-en-1-yl)amino]-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]benzamide
4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(trifluoromethyl)morpholine
2-{4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-[(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
2-[4-(1-benzylpiperidin-4-yl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
ethyl 5-{[(3-benzyl-4,5-dihydro-1,2-oxazol-5-yl)formamido]methyl}furan-2-carboxylate
5-(cyclopentylamino)-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-chloro-2-(4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidine
4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-ethyl-N-methylpiperidine-1-sulfonamide
(3S,4R)-3-methoxy-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-4-amine
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
N'-(3-chloro-4-fluorophenyl)-N-[2-(1H-imidazol-4-yl)ethyl]butanediamide
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-[(3-methylphenyl)methyl]piperidin-3-yl]propanoate
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}oxane-4-carboxamide
N-(3-fluorophenyl)-4-{2-[(2-methoxyethyl)carbamoyl]ethyl}piperidine-1-carboxamide
5-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-ethyl-1H-1,2,4-triazole
N-methyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine-3-carboxamide
2-(methylsulfanyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidin-4-yl}methanesulfonamide
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]pyridine
1-benzyl-8-(2,2-dimethylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-benzyl-1H-pyrazole-4-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine