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(3R,4S)-4-propyl-1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-amine
methyl 5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
9-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-9-(6-methylpyridine-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
(2S,4R)-1-(1H-imidazol-4-ylmethyl)-N-methyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)amino]pyrrolidine-2-carboxamide
methyl 2-({[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}(oxolan-2-ylmethyl)sulfamoyl)benzoate
{1-[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-3-ylmethyl)amine
2-{4-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]morpholin-3-yl}-N-methylacetamide
5-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-[2-(pyrrolidine-1-sulfonyl)ethyl]-3-(1,2,3-thiadiazol-5-yl)urea
[1-(4-aminopyrimidin-2-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
1-ethyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-3-ethyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
7-(cyclobutylmethyl)-2-(1-propylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane
2-(4-{[(4-chloro-3-methylphenyl)carbamoyl]amino}piperidin-1-yl)-N-cyclopropylacetamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]piperidine-1-carboxamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
7-[(2,3-dimethoxyphenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decane
(1S,5R)-6-(cyclobutylmethyl)-3-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(3-methoxyphenyl)-N-methylpropanamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyrrolidin-3-yl)benzamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(2-methylpropyl)-8-[2-(methylsulfanyl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-3-[4-(4-methylphenoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyrazin-2-yl)ethan-1-one
2-(cyclopropylmethyl)-N,7-dimethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2-oxa-7-azaspiro[4.5]decane
N-(4-fluoro-3-methylphenyl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-(3-fluorophenoxymethyl)-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-amino-3-ethyl-N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-4-(pyrrolidine-1-carbonyl)piperidine
3-(dimethylamino)-N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
(4aS,8aR)-1-(2-aminoethyl)-6-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(pyridin-2-ylmethyl)acetamide
(2S,4S)-4-amino-1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
{1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-2-yl}methanol
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1,7-dimethyl-1H-indole-2-carboxamide
2-(1H-1,3-benzodiazol-2-yl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
1-(3-chlorophenyl)-4-(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperazine
[(4-fluoro-3-methoxyphenyl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
2-({4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
ethyl 3-[(3-chlorophenyl)methyl]-1-(2,6-dimethylpyrimidine-4-carbonyl)piperidine-3-carboxylate
(3S,4R)-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
S-(4-{2-azaspiro[4.4]nonane-2-carbonyl}phenyl)-2-hydroxypropane-1-sulfonamido
(3aR,6aR)-2-benzyl-N-[2-(1H-pyrazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl 1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)azepan-4-yl]piperidine-4-carboxylate
(2R,6R)-1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine