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2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
4-(2,4-difluorophenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(dimethylamino)-4-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
N-[(3R,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-propyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
2-{5-[(dimethylamino)(3-fluorophenyl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-(5-chloro-1H-indole-2-carbonyl)-4-methyl-1,4-diazepan-6-ol
N-cyclopropyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(cyclohexylmethyl)-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
6-[3-(2-methylphenoxy)azetidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-(3-chloro-4-methylphenyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(2E)-3-(3-chlorophenyl)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
1-[(2-methoxyphenyl)methyl]-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-oxopiperidine-3-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(methylsulfanyl)ethyl]acetamide
1-[(diethylcarbamoyl)methyl]-N-[(2-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[4-(1H-1,3-benzodiazol-1-yl)-2-methoxyphenyl]acetamide
N-(2,4-dimethylphenyl)-3-{[1-(hydroxymethyl)cyclopentyl]amino}propanamide
2-(1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-3-carbonyl)pyridine
4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N,N-dimethyl-2-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamido]propanamide
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-3-fluorobenzamide
3-(1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(pyrrolidine-1-carbonyl)pyridine
3-(3-cyclobutyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)benzoic acid
1-[4-(3-methylphenoxy)piperidin-1-yl]-4-(morpholin-4-yl)pentan-1-one
3,3-dimethyl-1-({5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-4-(1H-imidazol-2-yl)piperidine
5-(4-ethyl-2-methyl-1,3-thiazol-5-yl)-3-methyl-1H-1,2,4-triazole
N-[3-(1H-imidazol-1-yl)propyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
2-cyclopentyl-N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)acetamide
3-[2-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-oxoethyl]-6-methoxy-2,3-dihydro-1H-indol-2-one
3-[1-(piperidine-1-sulfonyl)piperidin-3-yl]benzoic acid
2-amino-3-ethyl-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2R)-1-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)propan-2-ol
1-{[5-(azetidin-1-ylmethyl)-2,4-dimethylphenyl]methyl}-4-methylpiperazine
2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-4-(pyrazin-2-yl)phenol
(3-cyclopentylpropyl)({[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
1-(2-methoxyethyl)-3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1-(pyridin-2-ylmethyl)urea
1-(2-aminoethyl)-N-[1-(thian-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
methyl 7-oxo-9-(pyridin-3-ylmethoxy)-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[1-({1-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
4-benzyl-3-[2-(2,2-diethylmorpholin-4-yl)-2-oxoethyl]piperazin-2-one
1-(3-chlorophenyl)-4-[1-(cyclopentylmethyl)piperidin-3-yl]piperazine
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
5-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-ethyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
(1S,6R)-9-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-3,9-diazabicyclo[4.2.1]nonane