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1-{3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)amine
5-[2-(3-fluorophenyl)piperidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
(4S)-N-[(2,4-dichlorophenyl)methyl]-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-[(2,3,4-trifluorophenyl)methyl]pyrrolidine-3-carboxylic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-{5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)piperidin-2-one
1'-(3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanoyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-{1-[2-(5-acetylthiophen-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
5-(2,5-dimethylfuran-3-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,4-triazin-3-amine
4-hydroxy-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-hydroxybenzoyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
4-(prop-2-en-1-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}-N-(propan-2-yl)pyridine-4-carboxamide
4-methyl-2-(1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
4-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenyl)but-3-yn-1-ol
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2,3-dimethyl-1H-indole-5-carboxamide
1-(morpholin-4-yl)-3-{3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
[(2-fluorophenyl)methyl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
2-(ethylamino)-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-4-methyl-1,3-thiazole-5-carboxamide
1-(2-cycloheptylethyl)-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
5-(2-methoxyacetamido)-N,1-dimethyl-2-(pyridin-4-yl)-N-[1-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
6-cyclopentyl-N-[5-(dimethylamino)pentyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(3-hydroxyadamantan-1-yl)-1-(methoxymethyl)cyclobutane-1-carboxamide
1-[4-(2-methoxyphenyl)phenyl]-3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)urea
1-[1-({1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
5-fluoro-4-(pyrrolidin-1-yl)-2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrimidine
1-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
5-fluoro-2-[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]-1H-1,3-benzodiazole
1-benzyl-4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methyl-1H-1,2,3-triazole
1-methyl-2-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
6-methyl-2-({[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}methyl)quinolin-4-ol
N-[(4-fluorophenyl)methyl]-3-{1-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperidin-4-yl}propanamide
N-{1-oxaspiro[4.4]nonan-3-yl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-{3-[2-(2-hydroxyethyl)-3-oxo-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-6-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
8-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
[(3R,4S)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[(8-methoxyquinolin-2-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(morpholin-4-yl)-2-oxoacetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(1R,3S)-3-(2-aminoethoxy)-7-(5-methyl-1,3,4-thiadiazol-2-yl)-7-azaspiro[3.5]nonan-1-ol
2-methoxy-N-{3-[3-(1H-pyrazol-1-yl)butanamido]phenyl}benzamide
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
7-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one