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(3aR,6aR)-2-[(5-butylthiophen-2-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl({[1-(propan-2-yl)pyrrolidin-3-yl]methyl})[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-[4-(3,4-dimethylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
(2S,4S)-4-amino-N-methyl-1-(9-methyl-9H-carbazole-3-carbonyl)pyrrolidine-2-carboxamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
(2S,4S)-4-amino-1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
3-methyl-5-[1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
1-(2-{[(8-methoxyquinolin-2-yl)methyl](methyl)amino}ethyl)piperidin-2-one
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
(4S,4aS,8aS)-1-(oxane-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
(1R,5S)-N-{2-[(dimethylcarbamoyl)methyl]phenyl}-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-ethyl-7-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}(thiophen-2-ylmethyl)amino)butan-1-ol
4-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}benzoic acid
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[(3,5-dimethoxyphenyl)methyl]propanamide
N-[(2R,3R)-1'-(2-methyl-1,3-thiazole-4-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
5-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}sulfonyl)-1-propyl-1H-pyrazole
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(3-phenylpropyl)amine
N-[1-(1-cyclopentylpiperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N-methylthiophene-2-carboxamide
2-[(3-methoxyphenyl)sulfanyl]-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-[4-(2-fluoro-6-methoxyphenyl)phenoxy]-N-methylacetamide
N-(1-{7-[(4-acetamidophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N4-methyl-N2-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}pyrimidine-2,4-diamine
1-{4-[4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
1-cycloheptanecarbonyl-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-(2,2-diphenylethyl)-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
N-[(3S,4R)-1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-(furan-2-ylmethyl)-2-hydroxy-5-methyl-N-(prop-2-en-1-yl)benzamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)urea
2-{5-[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
4-[2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)ethyl]morpholine
ethyl 5-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-({1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-5-methylpyridine-3-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}oxolane-3-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-2-(propan-2-yloxy)-N-(pyridin-3-ylmethyl)propanamide
N-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-methyloxan-4-amine
N-(2-hydroxypropyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-[5-(morpholine-4-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
1-[1-(6-amino-2-methylpyrimidin-4-yl)piperidin-4-yl]piperidin-4-ol
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(pyridin-4-yl)piperazine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
N-(adamantan-1-yl)-2-{2-[(dimethylamino)methyl]-4-(pyrazin-2-yl)phenoxy}acetamide
(2S,4R)-4-(4-{[(cycloheptylcarbamoyl)amino]methyl}-1H-1,2,3-triazol-1-yl)-N-ethylpyrrolidine-2-carboxamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-(2,5-dimethoxyphenyl)-N-(2-methoxyethyl)acetamide
1-(2,3-difluorophenyl)-3-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
N-[(3R,4S)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
4-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]phenol