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1-(carbamoylmethyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(1-benzothiophen-2-ylmethyl)amino]-N-cyclopropyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
N3-[2-(quinolin-8-yloxy)ethyl]piperidine-1,3-dicarboxamide
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-8-fluoroquinolin-4-ol
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-N'-(2,4,6-trimethylphenyl)butanediamide
1-(3-fluorophenyl)-5-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidine-3-carboxamide
{9-[(3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
7-[2-(methylamino)pyrimidine-5-carbonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2-hydroxy-5-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(6-methylpyridine-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
2-(cyclohex-1-en-1-yl)-1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-hydroxyethyl)-N-propylpiperidine-3-carboxamide
4-chloro-2-{[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-2-(4-methyl-1,4-diazepane-1-carbonyl)pyrrolidin-1-yl]methyl}phenol
N-{2-[ethyl(methyl)amino]-2-methylpropyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(morpholin-4-ylmethyl)-1,4-oxazepane
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[1-(2-fluorophenyl)propan-2-yl]piperidine
2-[(1S,5R)-6-(1H-indazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-(4-methylphenyl)-N-[1-(pyrimidin-4-yl)ethyl]quinoline-4-carboxamide
5-fluoro-2-[1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-4-carboxamide
N-butyl-1,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{1-[3-(4-fluorophenyl)-3-oxopropyl]piperidin-3-yl}pyrrolidin-2-one
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
5-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-2-methylphenol
N-[3-(cyclohexyloxy)propyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
3-(3-chlorophenyl)-N-methyl-3-phenyl-N-(1,3-thiazol-2-ylmethyl)propanamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
(3aR,5R,6S,7aS)-2-(3-methoxybenzenesulfonyl)-octahydro-1H-isoindole-5,6-diol
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide
9-[(3-chloro-4-fluorophenyl)methyl]-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(4-{[3-methyl-1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
(butan-2-yl)({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-[(5-methylfuran-2-yl)methyl]piperidine-3-carboxylic acid
1-(4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-pyrazol-3-yl)-1H-1,2,3,4-tetrazole
7-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{3-[(2-fluorophenyl)methyl]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methanol
5-(4-fluorophenyl)-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-4-(ethanesulfonyl)phenol
1-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-5-phenylpentan-1-one
(5S,9aS,9bS)-2-(2-phenylethyl)-5-[3-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-(3-phenyl-1H-pyrazole-5-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine