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3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-(3-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)urea
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-benzothiophen-7-yl)-1-(cyclopropylmethyl)-6-{spiro[2.4]heptane-1-carbonyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(3-acetyl-1H-indol-1-yl)-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]butanamide
5-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
2-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
4-methoxy-N-methyl-3-({[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)benzamide
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
6-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methyl-1,2-dihydroquinolin-2-one
N-({7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
4-(hydroxymethyl)-1-[(6-methoxynaphthalen-2-yl)methyl]azepan-4-ol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(4-methyl-1H-imidazol-2-yl)methyl](oxolan-2-ylmethyl)amine
N-[(4-methoxyphenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)piperidin-1-yl]-2-methylpropan-1-one
1-cyclopropyl-N-methyl-6-oxo-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1-(1H-1,2,4-triazole-5-carbonyl)-1,2,3,6-tetrahydropyridine
2-(2-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
N-[3-(furan-2-yl)-3-phenylpropyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-methyl-1-(3-methylbutyl)-4-(quinolin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-phenyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-amine
4-(3-acetylbenzoyl)-1-(2-methylphenyl)piperazin-2-one
(3aS,6aS)-2-(2-methoxyethyl)-5-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-methoxypropan-1-one
3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-methyl-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-4-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)benzamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
1-{5-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]thiophen-2-yl}ethan-1-one
2-cyclopropanecarbonyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-N'-(4-methylphenyl)propanediamide
3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
1-(butan-2-yl)-N-ethyl-5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
methyl 3-benzamido-5-(cyclobutylamino)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-4-[(2-methylphenyl)sulfanyl]piperidine-1-carboxamide
2-(2,4-difluorophenoxy)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
2-(2-aminoethyl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]quinazolin-4-amine
1-cyclopentyl-N-ethyl-N-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aR)-5-[(5-chlorothiophen-2-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl}({[4-(trifluoromethyl)phenyl]methyl})amine
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
3-cyclopropyl-1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(1R,2R,6S,7S)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
[9-(1H-imidazol-2-ylmethyl)-3-(oxane-4-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
4-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-amino-8-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-cyclopentyl-1-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}methyl)urea