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2-{[2-(1-methanesulfonylpiperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
2-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-imidazole
3-(3-chlorophenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-3-phenylpropanamide
1-(2,6-dimethylpyridin-4-yl)-4-[3-(furan-2-yl)benzoyl]piperazine
(3R,4R)-4-[4-(2-phenylethyl)piperazin-1-yl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidin-3-ol
10-methoxy-5-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
N4-[2-(morpholin-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
5-tert-butyl-4-[(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)methyl]furan-2-carboxamide
2-(methylsulfanyl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
1-[(4-methoxyphenyl)methyl]-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
methyl 2-{8-[(3-hydroxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
N3-[(2,5-difluorophenyl)methyl]-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
(2R,3R,6R)-5-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-ethoxypropan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-N'-(2-methylphenyl)propanediamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-cyclopentylacetyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-[(2-chlorophenyl)methyl]-1-cyclohexanecarbonyl-1,4-diazepan-5-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
2-{[(2-methylphenyl)methyl]sulfanyl}-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
9-(4-aminopyrimidin-2-yl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[(3S,4R)-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
[(1-benzyl-1H-imidazol-2-yl)methyl](methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
1-[(2S,4R)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
7-(2-methoxyethyl)-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]pentan-1-ol
N-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
N,N,2-trimethyl-7-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3,3,3-trifluoro-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
5-cyclopropanecarbonyl-1'-(5-methylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-cyclopropyl-8-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
[4-benzyl-1-(2-ethylpyrimidine-5-carbonyl)piperazin-2-yl]methanol
3-[(3R,4S)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3R,4R)-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
3-(benzenesulfonyl)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-[(2R,3R)-1'-[(3-hydroxy-4-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-4-yl)propan-1-one
N-{2-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide