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2-cyclopropyl-4-hydroxy-N-[4-(pyridin-2-yl)butyl]pyrimidine-5-carboxamide
3,5-dimethyl-4-oxo-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
4-(4-methoxyphenyl)-2-methyl-N-(1-methyl-1H-indazol-5-yl)piperazine-1-carboxamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]azetidin-3-ol
2-{4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxylic acid
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](oxolan-2-ylmethyl)amine
2-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethoxy]ethan-1-ol
3-chloro-4-ethoxy-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]benzamide
(3R,4S)-4-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
(2S,4R)-4-(dimethylamino)-1-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxylic acid
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-indazol-1-yl)ethan-1-one
1-{[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
{2-[2-(2-chlorophenyl)-4-methylphenoxy]ethyl}(methyl)amine
3-[(4-fluorophenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
3-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-4-hydroxybenzonitrile
4-[1-(quinoline-8-carbonyl)piperidin-3-yl]benzoic acid
2-[5-(5-acetylthiophen-3-yl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]benzoic acid
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
N-ethyl-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
8-chloro-2-{[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[2-(4-fluorophenyl)ethyl]propanamide
N-(4-methoxy-3-{[(2,2,2-trifluoroethyl)carbamoyl]amino}phenyl)acetamide
[4-({1-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
(1S,4S)-2-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
5-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole
[(1-cyclopentylpiperidin-4-yl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
5-(2-fluorophenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
1-[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}pyrrolidine-3-carboxylic acid
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
N-[(2-chlorophenyl)methyl]-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}propanamide
2,6-dihydroxy-N-methyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
({4-[(1-cyclobutanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)(methyl)(naphthalen-1-ylmethyl)amine
(3S,4S)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
7-(cyclohexylmethyl)-2-(2-methoxypyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
1-(2,5-dimethylphenyl)-5-[1-(pyrrolidin-1-yl)propan-2-yl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-(oxolan-3-yl)-4-(pyrrolidin-1-yl)benzamide
1-(5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methylphenyl)-1H-pyrrole
9-[6-(morpholin-4-yl)pyrimidin-4-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide
N-cyclopentyl-2-methyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]methanol
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
1-{2-methyl-5-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
N-(1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide