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5,6-dimethyl-3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-3-yl}-5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidine
2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)-N-[(1R,2S)-2-phenylcyclohexyl]acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
{5-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-2-yl}methanol
N-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
2-(1-methyl-1H-pyrazol-4-yl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
3-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methyl-1,6-naphthyridine
N-cyclopentyl-5-[2-(3,4-dimethoxyphenyl)acetyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-1-yl)quinazoline
1-{2-oxo-2-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidin-1-yl]ethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-2-ethyl-N-(2-methoxyethyl)butanamide
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)ethan-1-one
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidine
1-cyclopentyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-oxopyrrolidine-3-carboxamide
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
1-(5-methanesulfonamido-2-methylphenyl)-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
[(3S,5R)-5-(hydroxymethyl)-1-({2-[(3-methoxyphenyl)methoxy]phenyl}methyl)piperidin-3-yl]methanol
N-[(3,4-dimethoxyphenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
8-fluoro-N-(2-hydroxyethyl)-4-oxo-N-(1,3-thiazol-2-ylmethyl)-1,4-dihydroquinoline-2-carboxamide
6-(2,6-dimethoxypyridin-3-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
8-{[4-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-cycloheptyl-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
N-[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-5-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]phenyl]acetamide
1-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]phenyl}pyrrolidin-2-one
N-(2-ethylphenyl)-2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoacetamide
4-(2,5-dihydro-1H-pyrrole-1-carbonyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole
4-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(5-ethoxyfuran-2-carbonyl)-2-[(3-fluorophenyl)methyl]morpholine
1-(cyclopropylmethyl)-N-ethyl-5-[2-(1H-imidazol-2-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethoxy)phenyl]propan-1-one
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}acetamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}propanamide
1-(3-methylbutyl)-8-(pyridin-2-ylmethyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}quinoxaline
ethyl 3-{[3-(4-methoxy-2-methylbenzoyl)piperidine-1-carbonyl]amino}propanoate
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-(propan-2-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S)-2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-3-phenylpropanoic acid
1-{1-[(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(2S,4R)-4-(dimethylamino)-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]pyrrolidine-2-carboxylic acid
2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1-methyl-1H-1,3-benzodiazole
(2S,4S)-4-cyclobutaneamido-1-(2,6-dimethylpyrimidine-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide