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N-cyclopentyl-N-[2-(dimethylamino)ethyl]-3-propanamidobenzamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(1-methoxypropan-2-yl)pyrimidin-2-amine
methyl 2-{1-[(3-methanesulfonamidophenyl)carbamoyl]pyrrolidin-3-yl}acetate
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(furan-2-carbonyl)piperazine
2-(4-fluorophenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-(2-chloro-4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetamide
methyl 4-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-1H-pyrazole-3-carboxylate
3-[3-(1H-pyrazol-3-yl)phenyl]benzonitrile
1-(2-{2-[2-(2-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)imidazolidin-2-one
3-[3-(phenoxymethyl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-4,6-dimethylpyrimidin-2-amine
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-(furan-2-ylmethyl)-2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-(2-benzamido-5-methylphenyl)-1H-pyrrole-2-carboxamide
2-cyclopentanecarbonyl-1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-methyl-6-{5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-1-yl}-1,3-benzothiazole
3-hexyl-8-[(2R)-2-hydroxy-2-phenylacetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({3-methyl-7-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
3-[4-(3-methylphenoxy)piperidin-1-yl]-5-(1H-pyrazol-4-yl)pyrazin-2-amine
(2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)urea
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
4-(cyclopropylmethyl)-1-{[2-(furan-2-yl)phenyl]methyl}-1,4-diazepan-5-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclohexanamine
5-{2-[(1-phenoxypropan-2-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine
4-{1-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]piperidin-3-yl}pyrimidine
4-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1-methylpiperazin-2-one
2-[({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)[(4-fluorophenyl)methyl]amino]butan-1-ol
2-cyclopropyl-N-ethyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
(2R,6S)-2,6-dimethyl-1-{[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
(2S)-N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-amino-3-(1H-imidazol-4-yl)propanamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-3-(2-methylfuran-3-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N,N-diethylpyrrolidine-2-carboxamide
N-[1-(1-{[(oxolan-2-ylmethyl)carbamoyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
8-(1-methyl-1H-pyrazole-4-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-(7-{[(2S)-2-(methoxycarbonyl)pyrrolidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidine-1-carboxylate
4-{[4-(cyclopentyloxy)phenyl]methyl}-1-(4-methoxyphenyl)piperazin-2-one
5-[(4-fluorophenyl)methyl]-5-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]acetamide
{2-[4-(adamantan-1-yl)piperazin-1-yl]quinolin-3-yl}methanol
4-[3-(2-chlorophenoxy)azetidin-1-yl]-5,6-dimethylpyrimidin-2-amine
3-(1-butyl-1H-imidazol-2-yl)-N-(2-methoxy-5-methylphenyl)piperidine-1-carboxamide
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-methoxyethyl)-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)propanamide
4-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-phenylpiperazin-2-one
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-(1-{[4-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
1-(cyclopropylmethyl)-N-methyl-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(5-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine