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{1-[1-(4-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}(methyl)(pyridin-2-ylmethyl)amine
2-[5-(2,5-dimethylfuran-3-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(3-phenylpropyl)piperidin-3-ol
2,3-dimethyl-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidine
4-[(4-fluorophenyl)methyl]-1-(4-methyl-1H-pyrrole-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-{[4-(hydroxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(2,3-dihydro-1H-inden-2-yl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
5-cyclopropyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
6-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(1-ethyl-3-oxopiperazin-2-yl)-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)acetamide
8-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-(5-propyl-1,2-oxazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]piperidine-4-carboxamide
1-(2-phenylethyl)-4-{[(trimethylpyrazin-2-yl)methyl]amino}pyrrolidin-2-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
1-(1-benzyl-1H-pyrazole-4-carbonyl)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
1-[2-(dimethylamino)ethyl]-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrrolidin-2-one
1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
(3S)-N,N-dimethyl-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}azepan-3-amine
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}piperidin-2-one
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1,4-diazepan-2-one
4-(3,5-dimethyl-1H-indole-2-carbonyl)-1-(3,5-dimethylphenyl)piperazin-2-one
N-butyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(azocan-1-yl)-N-[phenyl(pyridin-4-yl)methyl]propanamide
2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]benzonitrile
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(2-methoxy-5-methylphenyl)pyrazine-2-carboxylic acid
2-(2-chloro-4-{[2-(hydroxymethyl)azepan-1-yl]methyl}phenoxy)acetamide
N-cyclohexyl-3-[(furan-3-ylmethyl)sulfamoyl]-N-methylbenzamide
N-[2-(2-ethoxyphenoxy)ethyl]-N,2-dimethylimidazo[1,2-a]pyrimidine-3-carboxamide
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
2-(2,3-difluorophenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(cyclohex-1-en-1-yl)-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]propanamide
N-(oxolan-2-ylmethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(cyclopropylmethyl)-N-methyl-5-[3-(4-methylphenyl)propanoyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(4-methylphenoxy)piperidine
N-(pyridin-3-ylmethyl)-4-(1,3-thiazol-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(3,4-difluorophenoxymethyl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(pyridin-2-yl)propanoyl]piperidin-3-yl}propanamide
2-hydroxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-(1H-pyrrol-1-yl)benzamide
2-[2-(4-fluorophenyl)piperidine-1-carbonyl]benzonitrile
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-(4-methyl-1,4-diazepan-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-(azocan-1-yl)-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one