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5-[(isoquinolin-5-yloxy)methyl]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-{[3-(difluoromethoxy)phenyl]methyl}-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1,4-diazepan-6-ol
2,4-dimethyl-N-[1-(4-{[3-(morpholin-4-yl)propyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]benzamide
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methylfuran-3-carboxamide
N-(1-hydroxypropan-2-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-[(2R,3R)-2-ethoxy-1'-(1H-indole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
N,N-dimethyl-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
3-cyclohexyl-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)propanamide
8-fluoro-2-({[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)quinolin-4-ol
5-methoxy-2-[5-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
6-[(diethylamino)methyl]-N-(2-hydroxybutyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-methanesulfonylethan-1-one
9-methyl-2-{[2-(4-methylpentyl)morpholin-4-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-[(2E)-2-methylbut-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(3-fluorophenyl)-N-{1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]-1H-pyrazol-4-yl}acetamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2-(1,3-thiazol-2-yl)piperidine
4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}morpholine
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
1-(4-methanesulfonylphenyl)-2-(propan-2-yl)-1H-imidazole
4-{[4-methyl-5-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}morpholine
2-(4-chloro-2-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}phenoxy)acetic acid
2-methyl-8-(2-methyl-4-phenylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2,1-benzoxazole-3-carboxamide
(3R,4S)-N,N-dimethyl-1-(morpholine-4-sulfonyl)-4-propylpyrrolidin-3-amine
1-phenyl-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethane-1,2-dione
(8R,9aS)-2-{2-[(4-chlorophenyl)methoxy]ethyl}-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-{[3-methyl-7-(2-phenoxypropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
2-(1H-imidazol-2-yl)-N-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]benzamide
3-(2-chlorophenyl)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]-3-phenylpropanamide
N-(2-methoxyethyl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
(2R,6S)-1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2,6-dimethylpiperidine
2,5-difluoro-N-{1-[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
N-({7-[4-(methylsulfanyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
2,5-dioxo-6-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3S,4R)-4-(3-fluorophenyl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid
2-(dimethylamino)-N-{[4-(dimethylamino)-1-ethylpiperidin-4-yl]methyl}-2-(4-methylphenyl)acetamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
N,2-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzothiazole-5-carboxamide
methyl 3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 4-[3-(diphenylmethyl)-4,5-dihydro-1,2-oxazole-5-amido]piperidine-1-carboxylate
N-[2-(4,5,6,7-tetrahydro-1H-indazol-3-ylformamido)ethyl]pyridine-3-carboxamide
1-(1,3-benzoxazol-2-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid