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1-benzyl-5-methanesulfonamido-N,2-dimethyl-N-(thiophen-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
3-cyclohexyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
4-(4-chlorobenzoyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(cyclopropylmethyl)-N-ethyl-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
(2S)-2-acetamido-3-[1-(5-methylthiophen-2-yl)-1H-imidazol-4-yl]propanoic acid
N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-[4-(2-chlorophenyl)piperazin-1-yl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-propyl-1,2,3-thiadiazole-5-carboxamide
3-{2-oxo-2-[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
6-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-2-methyl-1,3-benzoxazole
8-fluoro-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
6-methyl-5-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-[2-(benzenesulfonyl)ethyl]-5-[4-(4-fluorophenyl)piperazin-1-yl]azepan-2-one
2-(furan-2-yl)-5-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrimidine
1-(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)-2-phenylethan-1-one
2-cyclopropyl-8-[2-(3,4-dimethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(1-methylpiperidin-4-yl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
(1S,6R)-9-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrazine
1-(2,3-dihydro-1H-inden-2-yl)-N-(thiophen-3-ylmethyl)piperidin-3-amine
N,N-dimethyl-4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-oxobutanamide
2-[(2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(2-fluorophenyl)methyl]-1,4-diazepane
2-[4-(4-fluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
8-[2-(2-methoxy-4-methylphenoxy)ethyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-(methylamino)-N-[(3R,4S)-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[(2-methoxynaphthalen-1-yl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
3-amino-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidine-3-carboxylic acid
2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}quinoline-4-carboxylic acid
1-[(2,6-difluorophenyl)methyl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-(3-benzoylpiperidin-1-yl)-2-(3-chlorophenyl)ethan-1-one
(1R,5R)-3-methanesulfonyl-6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-(1H-imidazol-2-yl)ethyl]-2-(2,4,5-trimethoxyphenyl)-1H-imidazole
(1S,5R)-3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2,3-dimethyl-6-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-(5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
6-(3-cyclopropyl-1-methyl-1H-1,2,4-triazol-5-yl)quinoline
N-cyclohexyl-2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methylacetamide
(2-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}ethyl)dimethylamine
5-(3-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}phenoxy)-1-azabicyclo[3.2.1]octane
(4aS,7aR)-N-(furan-2-ylmethyl)-4-(3-methylbutanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-(cyclopropylmethyl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
methyl(2-phenoxyethyl){[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}amine